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8-(1-benzofuran-2-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,3S,6R)-5-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-phenyl-5-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]pyrimidin-2-amine
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[1-(pyridin-3-yl)propyl]propanamide
(1R,5R)-3-cyclobutanecarbonyl-6-[(4-methanesulfonylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2-hydroxyethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(1,4-oxazepane-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[(3-chlorophenyl)methyl]-N-cyclopropyl-4-(piperidin-3-yl)benzamide
9-(2-amino-6-methylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-(6-methoxypyridin-3-yl)-2-(1,3-thiazol-2-yl)piperidine-1-carboxamide
2-{4-[(4-chlorophenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
1-cyclohexyl-5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-phenyl-N-({7-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
3-(diphenylmethyl)-N-(quinolin-3-ylmethyl)-1,2-oxazole-5-carboxamide
4-(4-methoxyphenyl)-6-methyl-2-oxo-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-N-phenylpropanamide
6-(1-benzofuran-2-yl)-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]pyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-5-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
5-[4-(cyclopropylmethyl)piperazine-1-carbonyl]-2-(2-phenylethyl)-1,3-benzoxazole
3-methyl-1-propyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
methyl 3-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)formamido]propanoate
5-cyclopropyl-N-(2-hydroxybutyl)-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
7-chloro-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1-(2-phenylethyl)-1,2-dihydroquinolin-2-one
3-[({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-1-methyl-1,2-dihydroquinolin-2-one
N,N-diethyl-2-({4-[2-(2H-indazol-2-yl)acetyl]-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl}oxy)acetamide
(1R,5R)-N-(4-chloro-2-methylphenyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-{[7-(3-cyclopentylpropanoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
1-[(2-methoxyphenyl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
methyl 4-oxo-4-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}butanoate
5-methyl-N-[4-(2-{[methyl(propan-2-yl)amino]methyl}propanamido)phenyl]furan-3-carboxamide
N-methyl-N-{2-phenyl-1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]ethyl}thiophene-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-N-{[7-(methylsulfanyl)-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}thiophene-2-carboxamide
N-[2-(dimethylamino)ethyl]-5-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1R,5R)-6-(cyclopropylmethyl)-N-(3,4-dimethoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-{3-[(2-phenylethyl)carbamoyl]piperidin-1-yl}-N-(prop-2-en-1-yl)piperidine-1-carboxamide
2-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-[(4-fluorophenyl)methyl]-4-[2-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-2-one
N-(1,4-oxazepan-6-ylmethyl)-5-(piperidine-1-carbonyl)pyridin-2-amine
(2R)-2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-4-methylpentanamide
3-cyclopropyl-5-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-methoxy-4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-cyclopropylacetamide
3-amino-N-(5-oxo-1-propylpyrrolidin-3-yl)-1H-1,2,4-triazole-5-carboxamide
3-(1-ethyl-1H-imidazol-2-yl)-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
5-(3-methoxyphenoxymethyl)-N-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
6-(4-methyl-1,3-oxazole-5-carbonyl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
N-(1-methyl-5-oxopyrrolidin-3-yl)-2-{5-[morpholin-4-yl(phenyl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-(methoxymethyl)furan-2-carboxamide
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-2-[3-(pyridin-2-yloxy)piperidin-1-yl]pyrimidine