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N-{2-[(4-chlorophenyl)methoxy]ethyl}-1-cyclopropanecarbonylpiperidine-4-carboxamide
1-(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidin-1-yl)-2-(pyridin-3-yl)ethane-1,2-dione
4-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-methylpiperazin-2-one
methyl 6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carboxylate
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]quinoxaline-6-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
3-(3-hydroxy-3-methylbutyl)-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)benzamide
3-[2-(dimethylamino)ethyl]-1-ethyl-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5S)-5-({[(2-methoxy-3,5-dimethylphenyl)methyl](pyridin-2-ylmethyl)amino}methyl)pyrrolidin-2-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(3-phenylpropyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
6-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinoline
1-[2-methoxy-2-(thiophen-2-yl)ethyl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
5-ethyl-5-{1-[3-(2-oxoazepan-1-yl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
N4-ethyl-N2,N4-dimethyl-N2-[2-(pyrrolidin-1-yl)ethyl]pyrimidine-2,4-diamine
4-methyl-3-[4-(2-methylpropyl)-1,4-diazepane-1-carbonyl]benzene-1-sulfonamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-[2-(4-methylpiperidin-1-yl)ethyl]-2-(methylsulfanyl)-N-(propan-2-yl)acetamide
N-{[3-methyl-7-(1-methyl-1H-indole-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
1-[4-({3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
3-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-amino-4-{4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
2-ethyl-1-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
N-[2-hydroxy-3-(4-methoxyphenoxy)propyl]-3-phenyl-1H-pyrazole-4-carboxamide
N-methyl-6-(piperidin-3-ylmethyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-1-{spiro[indene-1,4'-piperidine]-1'-yl}ethan-1-one
4-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
1-[3-(morpholin-4-yl)piperidin-1-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
(3S)-1-{2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}pyrrolidin-3-ol
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(3-phenylbutyl)benzamide
N-[3-(1H-imidazol-1-yl)propyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-(2-methoxy-2-methylpropyl)acetamide
N-ethyl-5-[1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)pyrrolidin-2-yl]thiophene-2-carboxamide
3-{2-[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-1-methylpiperidine
8-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(2,3-dimethoxyphenyl)ethyl]-4-(1H-1,2,4-triazol-3-yl)benzamide
1-ethyl-8-(2-ethylbutyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
methyl 1-{1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carbonyl}piperidine-4-carboxylate
1-[(2-methoxyphenyl)methyl]-N3-[(5-methylfuran-2-yl)methyl]-N5-[2-(methylsulfanyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-cyclohexyl-4-(dimethyl-1,3-thiazole-5-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
5-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidin-3-yl}-3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazole
N-(quinolin-4-ylmethyl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(1S,3R)-N1-[2-(furan-2-yl)ethyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
(3aS,6aR)-5-(3,6-dimethylpyrazin-2-yl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(2-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
N-cyclohexyl-3-[(6-hydroxy-1,4-oxazepan-4-yl)sulfonyl]benzamide
(3S,4R)-1-{[4-(difluoromethoxy)phenyl]methyl}-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
3-(2-methoxyphenyl)-1-methyl-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
(5S,9aS,9bS)-2-(2-phenylethyl)-5-(quinolin-8-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one