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2-methyl-6-{[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]amino}heptan-2-ol
4-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-(propan-2-yl)-1H-pyrazole
2-{4-[1-(oxan-4-yl)piperidine-3-carbonyl]piperazin-1-yl}pyrimidine
N-[2-(pyridin-3-yl)ethyl]-4-(pyrrolidin-1-yl)benzamide
N-({1-[(2H-1,3-benzodioxol-5-yl)carbamoyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
2-[(adamantan-1-ylmethyl)[(4-methyl-1H-imidazol-5-yl)methyl]amino]ethan-1-ol
N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-amino-N-ethyl-4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
(2S,4R)-4-amino-1-[2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1'-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}spiro[indene-1,4'-piperidine]
methyl 2-{5-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetate
3-[(4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidin-5-yl)formamido]-N-(1,3-thiazol-2-yl)propanamide
2-methoxy-N-[7-(4-methoxypiperidine-1-carbonyl)-1-(2-phenylethyl)-1H-1,3-benzodiazol-5-yl]acetamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(4-methyl-1,3-thiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-[5-(2-methanesulfonylethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]benzoic acid
8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methoxyethyl)-3-methyl-4-({[2-(pyrazin-2-yl)ethyl]carbamoyl}amino)benzamide
N-[2-(oxolan-3-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[2-(4-chlorophenoxy)ethyl]-3-(hydroxymethyl)piperidin-3-ol
N,N,4-trimethyl-3-({[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
10-(thiomorpholine-4-carbonyl)-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
[(2-methoxyphenyl)methyl][(6-methoxypyridin-3-yl)methyl](pyridin-3-ylmethyl)amine
2-cyclopropyl-1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1H-imidazole
N-ethyl-5-(methoxymethyl)-N-[2-(4-methoxyphenoxy)ethyl]furan-2-carboxamide
2-{[1-(1-benzyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]oxy}pyrimidine
7-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-6-carboxamide
1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(piperazin-1-yl)ethan-1-one
1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-{1-[(2-fluorophenyl)methyl]-4-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
4-(3-methylphenoxy)-1-(morpholine-4-carbonyl)piperidine-4-carboxylic acid
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
1-(2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenol
1-(4-acetylpiperazin-1-yl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethan-1-one
1-(2,3-dimethoxyphenyl)-2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-3-(2,5-dimethoxyphenyl)pyrrolidine-1-carboxamide
2-{5-[3-(benzyloxy)propyl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
7-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl](pyridin-4-ylmethyl)amine
3-(3-hydroxy-3-methylbutyl)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]benzamide
1-(1-benzoylpiperidin-4-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
2-[1-cyclopentyl-4-(2-ethylbutyl)piperazin-2-yl]ethan-1-ol
(4aR,7aS)-1-(1H-imidazol-4-ylmethyl)-4-(6-methoxyhexanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4-{[1-(furan-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
4-[2-(4-methoxyphenyl)ethyl]-3-(2-methyl-1,3-oxazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(1H-1,3-benzodiazol-1-yl)propyl]-N,1-dimethylpiperidin-4-amine
(1S)-2-({1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}amino)-1-phenylethan-1-ol
3-(2H-1,3-benzodioxole-5-carbonyl)-1-(1-benzyl-1H-pyrazole-4-carbonyl)piperidine
1-(9H-fluoren-2-ylmethyl)-4-(hydroxymethyl)azepan-4-ol