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3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-3-(2-methoxyphenyl)-1-(3-methoxypropyl)pyrrolidine-2,5-dione
1-(4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
methyl 3-(4-methyl-1,3-oxazole-5-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanamide
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-{[3-(methylsulfanyl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-(2-fluorophenoxymethyl)piperidine
2-[4-methoxy-3-(8-methoxy-2-methylquinolin-5-yl)phenyl]ethan-1-amine
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazole
methyl 2-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
3-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-1-{3-[(1-methylpiperidin-4-yl)oxy]propyl}urea
1-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazole
2-cyclopropylmethanesulfonyl-5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1-(2-methoxyethyl)-1H-imidazole
6-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidine-1-carbonyl)-2,3,4,9-tetrahydro-1H-carbazole
methyl 3-(1,3-benzothiazol-2-ylmethyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(6-cyclopropylpyrimidin-4-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
3-(piperidin-4-ylmethyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]benzamide
3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-(1,3-thiazol-4-ylmethyl)piperidin-4-ol
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-(methoxymethyl)cyclopropane-1-carboxamide
1-[4-(propan-2-yl)piperazin-1-yl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propan-1-one
6-methyl-4-(3,4,5-trimethoxyphenyl)-2,3-dihydropyridazin-3-one
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
4-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)piperazine-1-carbaldehyde
N-[2-(dimethylamino)-2-(4-methylphenyl)ethyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-({7-[2-(2-chloro-4-fluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
3-ethyl-8-[2-(1H-indol-3-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{[1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}azepan-2-one
3-(piperidin-1-ylmethyl)-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]propanamide
N-[2-(3-chlorophenyl)ethyl]-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
ethyl 2-[1-(2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)cyclohexyl]acetate
(1R,3S,5S)-8-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-8-azabicyclo[3.2.1]octan-3-ol
5-methyl-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}pyrazine-2-carboxamide
3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]-N-[2-(piperidin-1-yl)ethyl]propanamide
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,6,8-trimethylquinoline
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
N-(1-cyclopropanecarbonylpiperidin-3-yl)-2,6,8-trimethylquinoline-4-carboxamide
N-[(3-chlorophenyl)methyl]-3-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-4-yl]propanamide
5-{3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-(naphthalen-1-ylmethyl)pyrrolidin-2-one
N,N-bis(1,3-oxazol-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
methyl 5-[(2-{3',5',6',7'-tetrahydrospiro[cyclohexane-1,4'-imidazo[4,5-c]pyridine]-5'-yl}acetamido)methyl]furan-2-carboxylate
N-butyl-2,3-dimethyl-5-oxo-N-(thiophen-3-ylmethyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
4-(2,3-dihydro-1-benzofuran-2-carbonyl)-6-methyl-1-(2-methylphenyl)piperazin-2-one
3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)-5-{1-[2-(thiophen-2-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
N-butyl-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
5-(3-chlorophenyl)-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1,2,4-triazin-3-amine
3-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-N,N-dimethylaniline
N-(pyridin-2-ylmethyl)-3-[(thiolan-3-yl)sulfamoyl]benzamide