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1-(2-methoxyethyl)-5-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
(3S,4S)-4-cyclopropyl-1-(2,3-dichlorobenzoyl)pyrrolidine-3-carboxylic acid
N-(3-{4-[(cyclopropylformamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-5-methylthiophene-2-carboxamide
N-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
3-(furan-2-yl)-2-{2-[4-(methoxycarbonyl)phenyl]-1H-imidazol-1-yl}propanoic acid
7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(2R,3S,6R)-3-(4-methylphenyl)-5-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{1-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]piperidin-4-yl}-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
methyl (2S)-2-({7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazol-5-yl}formamido)-3-methylbutanoate
N-[3-(1H-imidazol-1-yl)propyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-methyl-N-(pyridin-3-ylmethyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
[1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-3-ethylpiperidin-3-yl]methanol
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
1-[6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl]-3-phenoxypropan-1-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,5-dimethyl-1,2-oxazole-4-sulfonamide
4-{1-[1-(3,5-dimethylphenyl)piperidin-4-yl]azetidin-3-yl}pyridine
2-(4-{[3-(furan-2-yl)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
1-(4-fluorophenyl)-N,6,6-trimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-methanesulfonyl-N-[2-(1H-pyrazol-1-yl)phenyl]piperazine-1-carboxamide
3-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1,2-benzothiazole
2-(4-ethylpiperazin-1-yl)-1-(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)ethan-1-one
2-methyl-5-oxo-N-[2-(propylsulfanyl)phenyl]-1,4-diazepane-1-carboxamide
4-[4-(1H-imidazol-1-ylmethyl)phenyl]benzamide
6-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-phenyl-4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
1-(oxan-4-yl)-3-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidine
1-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-(propan-2-yl)-2-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)acetamide
(3S,5S)-1-[2-(propan-2-ylsulfanyl)acetyl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3,5-dimethoxybenzamide
4-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}pyrimidine
9-[(2S)-2-aminopentanoyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]-2-methoxyacetamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
2,3,4-trimethoxy-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
4-[4-(1-methoxyethyl)phenyl]-2-methyl-5H,6H,7H-cyclopenta[d]pyrimidine
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
3-[(3R,4S)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-(1-ethylpiperidin-4-yl)-1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
(2S,4R)-4-amino-N-methyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidine-2-carboxamide
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-methoxy-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(2-fluoro-5-methanesulfonamidophenyl)urea
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-hydroxyacetamide
N-(4-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}phenyl)ethane-1-sulfonamide