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5-cyclobutyl-3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[2-(oxan-4-yl)ethyl]pyridin-2-amine
N-(2,2-difluoroethyl)-4-({[1-(methoxymethyl)cyclopropyl]methyl}sulfamoyl)benzamide
2-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-6,8-dimethylquinolin-4-ol
1-[4-(4-methoxyphenyl)phenyl]-3-{2-[(2R)-pyrrolidin-2-yl]ethyl}urea
4-[2-(dimethylamino)benzoyl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
1-[4-chloro-2-(trifluoromethyl)phenyl]-3-(pyrrolidin-3-yl)urea
(4aR,7aS)-1-(3-methylbutanoyl)-4-[(5-propylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{2-[4-(3-fluorophenoxy)piperidin-1-yl]ethyl}-1H-indazole
[2-(azepan-1-yl)ethyl](ethyl)(pyridin-4-ylmethyl)amine
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(4-methoxyphenyl)-3-phenyl-N-(pyridin-4-ylmethyl)propanamide
(3aR,6aR)-2-(2-acetamido-2-methylpropanoyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-methylpropyl)acetamide
2-(2-methoxyethoxy)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl 3-(4-{4-[(2-chlorophenyl)methyl]-2,5-dioxoimidazolidin-4-yl}piperidine-1-carbonyl)benzoate
3-[(cyclohexylamino)methyl]-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-[4-(3-methoxyphenyl)phenyl]-1-(1-propylpiperidin-4-yl)piperidine-3-carboxamide
2,4-dichloro-3-{[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]methyl}phenol
3-(4-methoxyphenyl)-N-(1,2-oxazol-3-ylmethyl)-3-phenylpropanamide
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
6-tert-butyl-N-(furan-2-ylmethyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-(3-ethyl-1H-pyrazole-5-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-(2-chloro-5-methylphenyl)-1-[5-(morpholin-4-yl)pentyl]urea
2-methoxy-N-{1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
1-[2-methoxy-4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(2-methoxyethyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
3-{[4-(6-chloroquinolin-2-yl)piperazin-1-yl]methyl}benzonitrile
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2,3-dihydro-1H-inden-1-yl)acetamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2-fluorobenzoyl)piperidine-2-carboxamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2-(quinazolin-4-yloxy)acetamide
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methyl-1H-1,3-benzodiazole-6-carboxamide
ethyl 1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-(4,6-dimethylpyrimidin-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(dimethyl-1,3-thiazol-5-yl)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
3-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 4-{[(5-acetyl-2-ethoxyphenyl)carbamoyl]amino}piperidine-1-carboxylate
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]butan-1-one
methyl 2-{[5-(2-cyclopentylacetamido)-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazol-7-yl]formamido}acetate
3-(2-methyl-1,8-naphthyridine-3-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
4-methanesulfonyl-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzene-1-sulfonamide
1-({4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-{4-[3-(pyridin-3-yl)propanoyl]morpholin-3-yl}acetamide
N-(2-{5-methyl-4-[(2-methylpropanamido)methyl]-1,3-oxazol-2-yl}phenyl)benzamide
N-(2-methoxyethyl)-1-methyl-N-[(4-methylphenyl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-methyl-1H-imidazol-1-yl)propanamide
5-(1H-1,3-benzodiazol-2-ylmethyl)-1-benzyl-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-ethyl-8-[(4-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-propanoyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one