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N-(dicyclopropylmethyl)-2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methylacetamide
4-[9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carbonyl]benzonitrile
N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)-2-(trifluoromethyl)benzamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
N-{[3-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-4-oxo-N-(pyridin-2-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-oxo-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
7-(5-methylthiophen-2-yl)-4-(quinoxalin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
N-[(2,3-difluorophenyl)methyl]-7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-fluoro-4-methylbenzamide
2-(dimethylamino)-N-{3-methyl-1-[7-(pent-4-enoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
methyl 2-oxo-8-(3-phenylpropyl)-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
8-(3-methoxy-4-methylbenzoyl)-2,8-diazaspiro[4.5]decan-3-one
1-(2-{1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}ethyl)pyrrolidin-2-one
2-(2-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-(4-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H-1,2,3-triazol-1-yl)propane-1,2-diol
2-{1-[(5-tert-butyl-2-hydroxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
2-{[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]amino}-N-methylpyridine-4-carboxamide
3-(3-methoxyphenyl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1H-pyrazole-4-carboxamide
N-cyclopropyl-1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-4-(trifluoromethoxy)benzene-1-sulfonamide
3-{3-[(3-methoxyphenyl)methoxy]phenyl}-6-methylpyridazine
4,4,4-trifluoro-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}butanamide
methyl 5-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
5-(hydroxymethyl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}furan-2-carboxamide
N-[(3S,4R)-1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
(1R,9aR)-1-[({2-[(3-methylpyridin-2-yl)amino]ethyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
(2R,6R)-4-{2-[(dimethylcarbamoyl)amino]acetyl}-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-(but-2-yn-1-yl)-5-{1-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(quinolin-4-ylmethyl)acetamide
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(3-methylbenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({8-[2-(3,4-dimethoxyphenyl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)cyclohexanecarboxamide
5-(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidine-1-carbonyl)-4-methylpyrimidin-2-amine
ethyl 1-ethyl-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N5-[2-(4-fluorophenyl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-benzofuran-2-carboxamide
1-benzyl-3-(2-methoxyethyl)-8-[(2E)-2-methylbut-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-cycloheptylpiperidin-3-yl)-4-(2-oxopiperidin-1-yl)butanamide
2-(propan-2-yl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-benzoxazole-5-carboxamide
2-[(3-ethyl-4-methylpiperazin-1-yl)methyl]-3,5-dimethoxybenzoic acid
2-(2-cyclopropylacetyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(oxolan-2-ylmethyl)-2,2-diphenylacetamide
2-{1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-1,3-benzoxazole
2-{[(1S,3aS,6aS)-octahydropentalen-1-yl]amino}-N-methylpyridine-4-carboxamide
2-[({[1-(2-hydroxyethyl)piperidin-3-yl]methyl}amino)methyl]-5,8-dimethylquinolin-4-ol
1-[2-({[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
methyl 2-[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})carbamoyl]piperidine-1-carboxylate
8-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione