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(3ar,6ar)-N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(3S,5R)-5-(4-methylpiperazine-1-carbonyl)-1-[(6-methylpyridin-2-yl)methyl]piperidine-3-carboxylic acid
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(2,3,6-trimethylphenoxy)acetamide
4-ethyl-3-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-[(2-cyclopentyl-2-phenylacetamido)methyl]-5-[2-(1,3-thiazol-4-yl)acetamido]benzoate
1-[2-(piperidin-2-yl)ethyl]-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
10-[3-(dimethylamino)pyrrolidine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
ethyl 4-(1-{[4-(methoxycarbonyl)phenyl]methyl}piperidin-3-yl)piperazine-1-carboxylate
2-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]oxane-2-carboxamide
(3S)-3-({1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-yl}amino)azepan-2-one
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-{2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4,5,6,7-tetrahydro-2H-indazole
N-[(3S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]-2-{1H-pyrrolo[2,3-b]pyridin-1-yl}acetamide
4-(5-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1H-pyrazol-3-yl)phenol
N-(1-{1-[6-(dimethylamino)pyrimidin-4-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[(2-fluorophenyl)methyl]piperazin-2-yl)ethan-1-ol
methyl 7-oxo-3-(quinoxalin-5-ylmethyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-(4-methoxyphenyl)-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
1-cyclopentyl-3-(2-methylphenyl)-3-{2-oxo-2-[2-(pyridin-3-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
3-(dicyclopropylmethyl)-3H,4H-pyrido[2,3-d]pyrimidin-4-one
2-methoxy-N-{1-[1-(2-methoxyethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
2-chloro-N-{2-[(2-methyl-1-benzofuran-7-yl)formamido]ethyl}benzamide
1-(diphenylmethyl)-4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
2-[9-(2-cyclopentylacetyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
1-{7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-N-methylpyrrolidine-3-carboxamide
2-methyl-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1-benzofuran-5-carboxamide
N-cyclopropyl-4-[1-(3-methylbutyl)-1H-pyrazol-4-yl]benzamide
(1S,5R)-6-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3,3-dimethyl-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(morpholin-4-ylmethyl)piperidin-4-ol
8-(6-methylpyridazin-3-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-5-methylthiophene-2-carboxamide
8-(4-chloro-3-ethoxybenzenesulfonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
2-({1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}amino)pyridine-3-carboxamide
4-(2-chlorobenzoyl)-6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
1-(cyclohexylmethyl)-N,N-dimethyl-5-[(pyridin-4-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-methoxy-3-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinoxaline
1-[4-(4-fluorophenyl)oxane-4-carbonyl]-3-(1H-imidazol-1-ylmethyl)piperidine
(5S,9aS,9bS)-2-(2-methoxyphenyl)-5-[1-(3-methylphenyl)-1H-imidazol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-methyl-5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
2-{1-[(2-ethoxyphenyl)methyl]-4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
1-acetyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]piperazine-1-carboxamide
4-(5-fluoroquinolin-8-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
3-[(3-methyloxetan-3-yl)methyl]-1-(4-sulfamoylphenyl)urea
2-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)quinoxaline
2-(1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}piperidin-2-yl)ethan-1-ol
6-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2,3-dimethylquinoxaline