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N-[4-(5-methyl-4-{[(3-methyl-5,6-dihydro-1,4-dioxin-2-yl)formamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-3-carboxamide
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-({[4-(dimethylamino)phenyl]methyl}amino)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
4-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-6-methyl-2-propylpyrimidine
1-(6-{4-[(4-methylphenyl)methyl]piperazin-1-yl}pyridin-3-yl)ethan-1-one
ethyl 3-[(4-fluorophenyl)methyl]-1-(1-methyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)piperidine-3-carboxylate
N-cyclopropyl-3-{1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-4-yl}propanamide
(1R,5R)-6-{[2-(5-methylfuran-2-yl)phenyl]methyl}-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2-fluorophenyl)methyl]-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
5-{1-[(3-hydroxyphenyl)methyl]pyrrolidin-2-yl}-N-(5-methyl-4H-1,2,4-triazol-3-yl)thiophene-2-carboxamide
5-[1-(3-methylbutanoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-(cyclopropylmethyl)-1-[4-(4-methylpiperazin-1-yl)benzoyl]piperidine-3-carboxylic acid
4-(hydroxymethyl)-1-[(4-methoxy-5,6,7,8-tetrahydronaphthalen-1-yl)sulfonyl]piperidin-4-ol
(1S,5R)-3-(3-propyl-1H-pyrazole-5-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(3-methoxyphenyl)-2-[(trimethyl-1H-pyrazol-1-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
(2R,6R)-10-methoxy-4-(pyridin-4-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3,5-dichloro-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,4-dimethylbenzamide
(3aS,6aS)-3a-(hydroxymethyl)-N-[2-(piperidin-1-ylmethyl)phenyl]-octahydrocyclopenta[c]pyrrole-2-carboxamide
(3S,5R)-5-(4-methylpiperazine-1-carbonyl)-1-(pyridin-2-ylmethyl)piperidine-3-carboxylic acid
N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
4-(4-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
5-[(benzyloxy)methyl]-4-phenyl-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole
4-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}piperazin-2-one
3-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-methylpyridazine
3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]-2,6,6-trimethyl-1-propyl-4,5,6,7-tetrahydro-1H-indol-4-one
9-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-[(2-methoxyphenyl)methyl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-[ethyl(methyl)amino]-2-methylpropan-1-one
[1-(1-{[4-(benzyloxy)-3-methoxyphenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
7-(cyclopropylmethyl)-2-{[4-(methylsulfanyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-3-[5-(2-ethoxyacetyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
4-methoxy-2-{4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine
methyl (2R)-2-({5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]phenyl}formamido)propanoate
3-[2-(3-methoxyphenyl)ethyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(1-benzylpiperidin-4-yl)-N-(2-methoxy-2-methylpropyl)piperidine-3-carboxamide
4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
4-{[2-hydroxy-5-(pyrimidin-5-yl)phenyl]methyl}piperazine-1-carbaldehyde
N-{[1-(phenoxymethyl)cyclopropyl]methyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}propanamide
2-(3-methoxyphenoxy)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
(2E)-3-(4-fluorophenyl)-1-(3-{5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)prop-2-en-1-one
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}){[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(2-methoxyphenyl)ethyl]propanamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-ethoxy-5-(3-methyl-1H-pyrazol-1-yl)benzamide
6-{[3-methoxy-4-(propan-2-yloxy)phenyl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-cyclopentyl-4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-one
1-(oxolan-2-ylmethyl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(2-chlorophenyl)-N-[(5-methylpyrazin-2-yl)methyl]-3-phenylpropanamide