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methyl 1-benzyl-5-[(oxan-4-yl)amino]-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2,3-difluorophenoxymethyl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-1,3-oxazole-4-carboxamide
1-{[5-(4-methylphenyl)furan-2-yl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-ethyl-3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
2-{2-[(6,8-dimethoxy-4-methylquinolin-2-yl)amino]ethoxy}ethan-1-ol
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2-(1H-1,2,4-triazol-1-yl)benzamide
1-(2-{4-[3-(4-methylphenyl)propanoyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
5-(1-benzofuran-2-yl)-N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1,2,4-triazin-3-amine
2-(4-fluorophenyl)-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)acetamide
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2,2-dimethylpropanamide
3-(2-methylpiperidin-1-yl)-N-[4-(pyridin-3-yloxy)phenyl]azetidine-1-carboxamide
2-chloro-4-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
{3-[(2,4-difluorophenyl)methyl]-1-(2,5-dimethylpyrimidin-4-yl)piperidin-3-yl}methanol
2-{4-[(3,4-dimethoxyphenyl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]propanamide
4-fluoro-N-{[1-(1-phenylcyclopropanecarbonyl)piperidin-3-yl]methyl}benzamide
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4-sulfamoylbutanamide
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}benzamide
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-[1-(quinolin-6-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
2-ethyl-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
4-{2-[5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine
4-{5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]furan-2-yl}-2-methylbut-3-yn-2-ol
6-methoxy-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-(butane-2-sulfonyl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-(adamantan-1-yl)-1-{1,3-dioxo-2-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
4-(dimethyl-1,2-oxazole-4-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-(1-{3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidin-4-yl)-2-phenylethan-1-ol
1-(2-chlorobenzoyl)-4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
3-benzyl-8-{[3-(furan-2-yl)phenyl]methyl}-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-ethyl-2-methyl-1,3-thiazole-5-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(1H-pyrazol-1-yl)benzamide
2-(4-propyl-4H-1,2,4-triazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-3-yloxy)propyl]amine
ethyl 4-{3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanoyl}piperazine-1-carboxylate
3,5-difluoro-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyridine-2-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(furan-2-yl)-N-(oxolan-2-ylmethyl)propanamide
2-(3-fluorophenoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide
5-(2-cyclopentylacetamido)-N,1-dimethyl-2-(oxolan-2-yl)-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
(2S,4S)-4-[1-(4-chlorophenyl)cyclopropaneamido]-N-ethyl-1-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
2-{1-cyclopentyl-4-[(3-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-cyclopropyl-3-{5-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(4-fluorophenyl)piperidin-4-ol
methyl 2-(7-chloro-3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-2-oxo-1,2-dihydroquinolin-1-yl)acetate
N-(2-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
2-[(3-methoxyphenyl)methyl]-8-(oxolane-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(1-benzofuran-5-yl)-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazole
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
1-[5-methoxy-2-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol