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[(3R,4R)-1-[(2-chloro-3,6-difluorophenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-(4-chloro-1-propyl-1H-indazol-3-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide
5-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-4-propyl-1,2,3-thiadiazole
5-(piperidine-1-carbonyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
N3-butyl-N3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-1,3-dicarboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[(isoquinolin-5-yloxy)methyl]-N-methyl-1,2-oxazole-3-carboxamide
5-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indazole
8-{[4-(1,2-oxazolidine-2-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
N-[(2-chlorophenyl)methyl]-8-fluoro-N-(2-hydroxyethyl)quinoline-2-carboxamide
N-(butan-2-yl)-N-[(2-fluorophenyl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-(2-aminoethyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}quinazolin-4-amine
4-({4-methyl-5-[1-(1-methylcyclopentanecarbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-methyl-9-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2,4-dimethylbenzamide
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(1H-imidazol-1-yl)acetamide
1-[5-({[(2,4-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
2-[(5-methylpyrazin-2-yl)methyl]-8-(2-methylpyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
[2-(2-methoxyphenyl)ethyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-8-methyl-1,4-dihydroquinolin-4-one
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
2-(2-{1-[2-(2-methyl-1H-indol-3-yl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(4-methylphenyl)methyl]-2-(propan-2-yloxy)acetamide
2-(4-chlorophenyl)-4-{imidazo[1,2-a]pyridine-6-carbonyl}morpholine
N-[(3R,4R)-3-hydroxy-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidin-4-yl]pyridine-4-carboxamide
3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-(morpholin-4-yl)quinoline
N,N-dimethyl-2-[(1S,5R)-6-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
3-(2-cyclohexylacetyl)-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-3,4-dihydroquinazolin-4-one
5-(2,7,8-trimethylquinoline-4-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
N,N-diethyl-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carboxamide
2-{[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
1-benzyl-3-(2-methoxyethyl)-8-[(3-phenoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-ethyl-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidine-5-carboxamide
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1,1-dioxo-1λ6-thiolane-3-carboxamide
4-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
methyl (2S)-1-[9-methoxy-7-oxo-3-(2-phenoxyacetyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
1-(3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
N-[(2R,3R)-1'-(1-ethyl-1H-pyrazole-4-carbonyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
methyl 1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazole-4-carboxylate
methyl 3-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}benzoate
4-(1H-imidazol-1-yl)-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidine-4-carboxylic acid
N-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]oxan-4-amine
4-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]-2-methoxypyridine-3-carbonitrile
N-cyclopropyl-N-({4-methoxy-3-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)oxolane-2-carboxamide
N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-(2,3-dihydro-1H-inden-2-yl)-N-methylacetamide
5-{3-[3-(benzyloxy)piperidin-1-yl]-3-oxopropyl}-5-[(3,4-dimethoxyphenyl)methyl]pyrrolidin-2-one
3-[2-(cyclohex-1-en-1-yl)acetyl]-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-chloro-1-methyl-3-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)-1H-indazole