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4,6-dimethyl-2-oxo-N-[2-(pyridin-4-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
2-[2-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)phenoxy]propanoic acid
1-[(4-chlorophenyl)methyl]-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-{4-[(4-methylpiperazin-1-yl)sulfonyl]piperazin-1-yl}-4-(propan-2-yl)pyrimidine
8-chloro-2-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}quinoline
3-chloro-N-cyclopentyl-4-{[1-(2-methylpropanoyl)piperidin-4-yl]oxy}benzamide
3-(2-fluorophenoxy)-1-[3-(methylsulfanyl)propyl]azetidine
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)(3-phenylbutyl)amine
4-[5-(6-methylpyridazin-3-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
N-cyclopropyl-1-{1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(6-methylpyridin-2-yl)methyl]benzamide
(4aS,8aR)-6-(1,4-dimethyl-1H-indole-2-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-methanesulfonyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]pyrrolidine-2-carboxamide
3-(5-acetyl-2-ethoxyphenyl)-1-[3-(pyridin-3-yl)propyl]urea
2-(dimethyl-1,3-thiazol-5-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
1-{3-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
2-[8-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
N-(3-chloro-4-methoxyphenyl)-2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}ethan-1-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]piperidine-4-carboxamide
3,4-dimethoxy-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]benzene-1-sulfonamide
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-2-(trifluoromethoxy)benzene-1-sulfonamide
(2R,6R)-4-(1,4-dithiepan-6-yl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(dimethylamino)-7-[(3-hydroxy-4-methoxyphenyl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-{2-[6-(dimethylcarbamoyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamido}-2,2-dimethylpropanoic acid
1-[(3S,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-[(2R,3R)-1'-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-[2-({3-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}methyl)quinolin-6-yl]acetamide
3-[3-(1H-imidazol-2-yl)piperidin-1-yl]-6-phenylpyridazine
3-methanesulfonamido-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
(5S,9aS,9bS)-2-cyclopentyl-5-(3-hydroxy-4-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(4-phenylphenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
6-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-benzyl-3-ethyl-1-(5-methylpyrazine-2-carbonyl)-1,4-diazepan-5-one
(2S,4R)-4-(3,3-dimethylbutanamido)-N-methyl-1-(9H-purin-6-yl)pyrrolidine-2-carboxamide
N-[1-cyclopentyl-7-(3-methylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]benzamide
methyl 1-(2-methoxyethyl)-5-[(oxan-4-yl)amino]-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{1-[2-(azepan-1-yl)acetyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
1-(4-fluorophenyl)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,2-dimethylcyclopropane-1-carboxamide
1-[(4-chlorophenyl)methyl]-6-oxo-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidine-3-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)pyrazine-2-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
3-butyl-1-methyl-4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazin-2-one
N-[(2-methoxyphenyl)methyl]-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-propylacetamide
1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]-3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propan-1-one
7-[(3-methoxyphenyl)methyl]-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decane
[2-(4-methoxyphenyl)ethyl][(5-methylfuran-2-yl)methyl][(1-methylpiperidin-4-yl)methyl]amine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]pyrrolidin-3-yl]methanol
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]({[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-[2-(3-methoxyphenyl)ethyl]-5-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide