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5-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-phenyl-1H-imidazole
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
1-(cyclohexylmethyl)-3-hydroxy-3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
2-(3-cyclopropanecarbonyl-1H-indol-1-yl)-N-[(1-methylpyrrolidin-3-yl)methyl]acetamide
6-{3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
(3R,4R)-1-[2-(4-fluorophenoxy)ethyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylpropanamide
3-(3-fluoropyridin-4-yl)-4-methoxy-N-methylbenzamide
3-(methoxymethyl)-1-[(3,4,5-trimethoxyphenyl)methyl]pyrrolidine
N-[3-(1H-indazol-1-yl)propyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-ethyl-7-(2-methoxybenzamido)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methyl-1H-pyrazole-4-carboxamide
2-benzyl-4-(oxane-4-carbonyl)morpholine
N-[(3S,4R)-1-(2,4-dimethylpyrimidine-5-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
2-{2-[({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}pyrimidin-4-amine
[(4-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-2-yl}phenyl)methyl]dimethylamine
2-[2-(benzyloxy)phenyl]pyridine-4-carboxamide
8-(3-methoxypyrazin-2-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
3-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-1-(1,3,4-thiadiazol-2-yl)urea
N-benzyl-N-methyl-3-({[1-(propan-2-yl)piperidin-4-yl]amino}methyl)pyridin-2-amine
N-[2-(diethylamino)ethyl]-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-methylacetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-methoxy-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}benzamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-[1-(naphthalen-1-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
2-{4-[3-(azocan-1-yl)propanoyl]-3-methyl-2-oxopiperazin-1-yl}acetic acid
(4aS,8aR)-4a-(hydroxymethyl)-N-(2-phenylphenyl)-decahydro-1,6-naphthyridine-6-carboxamide
5-oxo-N-{[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyrrolidine-2-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
1-[2-(azetidin-1-ylmethyl)-6-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-[2-(pyridin-3-ylformamido)ethyl]benzamide
1-(cyclohexylmethyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-methoxyethyl)-8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-2-one
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
2-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-N,N-bis(prop-2-en-1-yl)acetamide
methyl 5-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-(3-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}propyl)-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-({5-[(2-phenoxyethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)cyclopropanecarboxamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
4-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1-methylimidazolidin-2-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-(4,5-dimethylthiophene-2-carbonyl)-4-[(4-fluorophenyl)methyl]-1,4-diazepane
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,1-benzoxazole-3-carboxamide
3-[(2-fluoro-5-methoxyphenyl)methyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}pyridine
1-ethyl-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrrolidin-2-one
5-[(benzyloxy)methyl]-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazole
4-({1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}methyl)morpholine