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2-{[(1,2-diphenylethyl)amino]methyl}-4-(pyrimidin-2-yl)phenol
ethyl 4-[3-({[(4-fluorophenyl)methyl]amino}methyl)-6,7-dimethoxyquinolin-2-yl]piperazine-1-carboxylate
ethyl 4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carboxylate
2-{2-[3-methyl-1-(2-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}acetamide
{[5-(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}methyl)cycloheptanecarboxamide
4-acetyl-6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one
9-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-3,9-diazaspiro[5.6]dodecane
N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-methyl-5-[3-(pyridin-4-yl)azetidine-1-carbonyl]-2,3-dihydro-1,3-benzoxazol-2-one
4-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-(quinolin-8-yl)-1,4-diazepane-1-carboxamide
3-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
1-[cyclohexyl(methyl)amino]-3-(2-{[(quinolin-6-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
(1S,5R)-6-(2-ethylpyridine-4-carbonyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(3,5-dimethoxyphenyl)methyl]-3,4-dihydropteridin-4-one
N-[(2R,3R)-1'-[(3,5-difluorophenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
{[(3S,4R)-1-[(2,5-dimethoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
(4aS,8aR)-1-(2-aminoethyl)-6-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-decahydro-1,6-naphthyridin-2-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-(4-{2-[cyclopentyl(methyl)amino]acetamido}phenyl)-5-methylfuran-3-carboxamide
3-methyl-N-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}pyridine-4-carboxamide
1-(1-{3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanoyl}piperidin-3-yl)-3-methylbutan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-phenyl-1H-pyrazole-4-carboxamide
1-{[2-(methylsulfanyl)phenyl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
1-{[5-(3-chloro-4-methylphenyl)furan-2-yl]methyl}-1,4-diazepane
2,3-difluoro-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
(1R,5S,8S)-3-[(4-chloro-3-fluorophenyl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
3,7-dimethyl-8-(4-methylthiophen-3-yl)-2,3,6,7-tetrahydro-1H-purine-2,6-dione
4-ethoxy-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyrimidine
(1S,9R)-11-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
6-(2-methoxyphenyl)-N-methyl-N-(thiophen-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
8-(cyclobutylmethyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(3-chlorophenyl)ethyl]-2-[(prop-2-yn-1-yl)amino]acetamide
(2R)-2-amino-3-(1H-indol-3-yl)-1-(4-phenyl-1,4-diazepan-1-yl)propan-1-one
2-(butylsulfanyl)-6-[3-(dimethylamino)pyrrolidin-1-yl]pyrimidin-4-amine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
6-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine-3-carboxylic acid
1-{5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-[(2R,3R)-2-methoxy-1'-(thiophene-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
2-methyl-6-[3-(5-methylfuran-2-yl)-1-propyl-1H-1,2,4-triazol-5-yl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
(3S,4R)-1-[(4-methoxy-3-methylphenyl)methyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
(2S,4S)-N-ethyl-4-(2-methoxyacetamido)-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidine-2-carboxamide
ethyl 5-[(3-hydroxyphenyl)methyl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]-2-(thiophen-3-yl)ethan-1-one
(2S,4S)-N-methyl-4-{4-[4-(1,2,3,6-tetrahydropyridin-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide