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5-(3-benzoylpiperidine-1-carbonyl)-2-cyclopropyl-3,4-dihydropyrimidin-4-one
N-[(2R,3R)-1'-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N-[2-(propylsulfanyl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]propanamide
3-(azepane-1-carbonyl)-N-(2-methoxyethyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1-cycloheptylpiperidin-3-yl)-4-(2-oxopyrrolidin-1-yl)butanamide
7-methyl-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]imidazo[1,2-a]pyridine-2-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-(3-fluorophenyl)-1,2,4-triazin-3-amine
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[3-(1H-1,2,4-triazol-1-yl)propyl]acetamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-amino-6-(3-fluoro-4-methoxyphenyl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
2-{4-[1-cyclohexyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}acetamide
4-{3-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperazin-2-one
2-({methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amino}methyl)phenol
2-methyl-6-{1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
2-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1-methyl-1H-1,3-benzodiazole
1-({4-[(2,4,5-trimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-4-ol
N-benzyl{[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]amino}sulfonamide
N-[3-({[2-(morpholin-4-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-4-(1H-pyrazol-1-ylmethyl)piperidine-1-carboxamide
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-5-propylimidazolidine-2,4-dione
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2,3-dihydro-1-benzofuran-7-carboxamide
1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-(4-methylphenoxymethyl)-1H-1,3-benzodiazole
3-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]urea
ethyl 1-(4-acetamidobenzoyl)-4-(2-methoxyethyl)piperidine-4-carboxylate
5-{[(2-chlorophenyl)methyl]amino}-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-hydroxyethyl)-1-[(1s,4s)-4-(cycloheptylamino)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridin-2-amine
methyl (1S,3S,3aR,6aS)-3-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-1-(hydroxymethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-(1H-indazol-7-yl)-4-[2-(morpholin-4-yl)ethyl]piperazine-1-carboxamide
4,6,7-trimethyl-2-{4-[4-(pyridin-3-yloxy)piperidin-1-yl]piperidin-1-yl}quinazoline
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}propanamide
1-(5-ethyl-1H-pyrrole-2-carbonyl)-3,3-diphenylpiperidine
N-(3,5-dimethoxyphenyl)-3-[1-(3-fluoro-4-methoxybenzoyl)piperidin-3-yl]propanamide
ethyl 5-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-({4-[(3,5-dimethoxyphenyl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]propanamide
6-ethyl-N,4-dimethyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]quinolin-2-amine
(1S,5R)-3-benzyl-6-(pyrrolidine-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[4-(4-fluoro-3-methoxyphenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]propanamide
1-(2,4-difluorophenyl)-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}urea
4-(1-{[4-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)morpholine
2-(2-phenylethyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]morpholine
3-(1H-pyrazol-1-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
4-(2-methoxyphenoxy)-1-(1-methylpiperidin-4-yl)piperidine-4-carboxylic acid
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-2-(2-phenylethyl)piperidine
N-benzyl-N-[2-(dimethylamino)ethyl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
2-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperazin-1-yl}ethan-1-ol
2-methyl-6-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)heptan-2-ol
N-ethyl-N-methyl-3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-sulfonamide
3-(1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,3-triazol-4-yl)piperidine