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3-[2-oxo-2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethyl]-1,2,3-oxadiazol-3-ium-5-olate
1-cyclobutanecarbonyl-4-(2,3-dihydro-1H-indene-1-carbonyl)-1,4-diazepane
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methanol
N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 3-[(2-methylphenyl)methyl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[2-(cyclopentylcarbamoyl)ethyl]-3-(cyclopropylmethyl)piperidine-3-carboxylic acid
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-fluorophenyl)methyl]piperidine
ethyl 2-({2,7-diazaspiro[4.5]decane-7-carbonyl}amino)benzoate
2-amino-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]hexan-1-one
1-[2-(dimethylamino)ethyl]-N-methyl-N-(naphthalen-1-ylmethyl)-5-oxopyrrolidine-3-carboxamide
(5-{1-[4-(pyridin-2-yl)butyl]-1H-imidazol-2-yl}furan-2-yl)methanol
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1-phenylcyclopropane-1-carboxamide
2-(4-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
2,6-dimethyl-N-[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]quinoline-3-carboxamide
2-methyl-6-({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)pyrimidin-4-ol
5-(methoxymethyl)-N-[(7-{[4-(pyrrolidin-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]furan-2-carboxamide
5-oxo-1-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrrolidine-3-carboxylic acid
N-[(2S,4R,6S)-2-(2,3-dimethoxyphenyl)-6-ethyloxan-4-yl]benzamide
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-(1-methyl-1H-indol-3-yl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-{4-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-1-yl}pyrazine
3-{cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}propane-1,2-diol
1-[4-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)phenyl]imidazolidin-2-one
(1R,2R,6S,7S)-4-(4-phenyl-1,3-thiazol-2-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-ethyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
1-ethyl-4-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperazine
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
3-(4-chloro-1H-pyrazol-1-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
1-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-{2,7-diazaspiro[4.5]decan-7-yl}-2-hydroxyethan-1-one
4-[(2-methoxypyridin-3-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
6-methoxy-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl 4-(4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
2-chloro-N-(2-{8-oxo-2-oxa-7-azaspiro[4.5]decan-7-yl}ethyl)benzamide
[(4-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-1,4-oxazepan-6-yl)methyl]dimethylamine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-methylazepane-2-carboxamide
{1-[(4-ethoxyphenyl)methyl]-3-[(4-fluorophenyl)methyl]piperidin-3-yl}methanol
1-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
2-(2-hydroxyphenyl)-1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}ethan-1-one
1-{4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-(1H-pyrazol-4-yl)propan-1-one
4-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-N-[(2S)-1-methoxypropan-2-yl]pyrimidin-2-amine
methyl 3-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}benzoate
ethyl 2-{[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]amino}acetate
1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-({[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
[5-(1-{1-oxaspiro[4.4]nonan-3-yl}-4-phenyl-1H-imidazol-5-yl)furan-2-yl]methanol
1-methyl-3-(2-methylpropyl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
ethyl 1-(2-methoxypyridine-3-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate