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N-(4-chloro-2-methoxy-5-methylphenyl)-4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazine-1-carboxamide
ethyl 2-[4-(5-chloro-3-cyano-4,6-dimethylpyridin-2-yl)piperazin-1-yl]acetate
5-oxo-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}phenol
N-butyl-2-(4-methylpiperazin-1-yl)-N-[(5-methylthiophen-2-yl)methyl]propanamide
2-[(4-methoxypyridin-2-yl)methyl]-1,2-dihydrophthalazin-1-one
3-(4-chlorophenyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-3-phenylpropanamide
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
2-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1'-[(2,6-difluoro-3-methylphenyl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-{[2-(3-methoxyphenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-[2-(4-benzoylpiperazin-1-yl)-2-oxoethyl]-4-(2-methylpropyl)pyrrolidin-2-one
(2E)-N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)prop-2-enamide
3-[(1-phenylcyclohexyl)methyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
3-{1-[1-(morpholin-4-yl)cyclohexanecarbonyl]piperidin-4-yl}-N-phenylpropanamide
methyl (2S,4R)-4-[3-(3-fluorophenyl)benzamido]-1-[(4-fluorophenyl)methyl]pyrrolidine-2-carboxylate
4-{4-[(4-ethyl-1,4-diazepan-1-yl)methyl]phenyl}but-3-yn-1-ol
N-butyl-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carboxamide
ethyl 4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine-1-carboxylate
4-(4-chlorophenyl)-1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-ol
4-(2-{[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]oxy}hex-5-en-1-yl)morpholine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-{[7-(2,4-difluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-3-(2-methoxyphenyl)-N-(pyridin-4-ylmethyl)propanamide
4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-1-(4-methylphenyl)piperazin-2-one
N-({7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
1-(3-methoxyphenyl)-4-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pyrrolidin-2-one
N-[2-(1,3-benzoxazol-2-yl)ethyl]-4-ethyl-5-methylpyrimidin-2-amine
2-[1-cyclohexyl-4-(isoquinolin-5-ylmethyl)piperazin-2-yl]ethan-1-ol
5-(3-methoxyphenoxymethyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylthiophene-2-carboxamide
1-(3-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S,4S)-1-benzyl-4-{[(2,4-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
(1R,7S)-N-methyl-4-oxo-3-[4-(propan-2-yl)phenyl]-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-[4-(oxolan-2-ylmethyl)piperazin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
7-chloro-4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-benzyl-3-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(3-methoxyphenyl)ethan-1-one
N-[(2-fluorophenyl)methyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-ethyl-N-methylacetamide
3-[4-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenyl]prop-2-yn-1-ol
(3S,4R)-1-(azepane-1-sulfonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-cyclobutanecarbonyl-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]imidazolidine-2,4-dione
(2S)-1-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidine-2-carboxamide
3-(3-methoxybenzoyl)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-1H-pyrazole-4-carboxamide
3-(5-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-2-yl)prop-2-yn-1-ol