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3-(3-fluorophenyl)-4-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]piperazin-2-one
1-[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]-3-methoxypiperidine
1-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3,3-bis(2-hydroxyethyl)urea
3-[(5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}furan-2-yl)sulfanyl]-4-methyl-4H-1,2,4-triazole
N-[(5-chloro-1H-indol-2-yl)methyl]-2,6-difluorobenzamide
1-cycloheptyl-N-methyl-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
(1S,5R)-3-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 3-(3-chlorobenzamido)-6-(morpholin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
2-(4-{furo[3,2-c]pyridin-4-yl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N,5-dimethyl-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(morpholin-4-yl)ethan-1-one
3-methoxy-N-(1-{7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-4-[3-(thiophen-2-yl)propanoyl]-1,4-diazepan-2-one
N-(1-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
N-{1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}acetamide
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
methyl 1-(3-{[4-(dimethylamino)phenyl]methyl}-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl)piperidine-2-carboxylate
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-6-(2,3,4-trimethoxyphenyl)pyridine-3-carbonitrile
N-cyclohexyl-3-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]propanamide
1-{[(3R,4R)-1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
5-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-5,6-dihydrophenanthridin-6-one
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-sulfonamide
2-[(3S,4S)-3-carboxy-4-(pyridin-2-yl)pyrrolidin-1-yl]-1,3-oxazole-4-carboxylic acid
(4aR,8aS)-1-[2-(3,4-dimethoxyphenyl)ethyl]-6-[3-(2-oxopyrrolidin-1-yl)benzoyl]-decahydro-1,6-naphthyridin-2-one
1-(5-fluoro-2-methylphenyl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
(2S,4R)-N-ethyl-1-[4-(hydroxymethyl)benzoyl]-4-[(3E)-pent-3-enamido]pyrrolidine-2-carboxamide
N3-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(cyclohexylmethyl)-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[4-(2-methoxyethyl)piperazin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
methyl (2S)-2-(3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamido)-3-methylbutanoate
(1R,7S)-3-tert-butyl-N-methyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]acetamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)-2-methoxypyridine
N-[2-(2,3-dimethoxyphenyl)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(2-methylpyrimidin-5-yl)methyl]piperidin-3-amine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(2-oxopyrrolidin-1-yl)propanamide
3-(2-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-1H-pyrrol-1-yl)benzonitrile
4-(1-benzylpiperidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[2-(piperazin-1-yl)ethyl]-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
2-(2-{1-[2-(3,4-dimethoxyphenyl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-[2-(dimethylamino)ethyl]-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-ethyl-1,7-dimethyl-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
5-[(2-methoxyethyl)amino]-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
9-methoxy-N-[(3-methoxyphenyl)methyl]-3-[(2-methylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-4-(morpholine-4-carbonyl)pyridin-2-amine
3-{4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-1H-indole
(3R,4R)-4-amino-1-[2-(phenylsulfanyl)ethyl]piperidin-3-ol
1-{[6-(1-benzofuran-2-yl)pyridin-3-yl]methyl}-4-methylpiperazine