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2-{[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
1-[(3-fluorophenyl)methyl]-4-(2-hydroxy-4-methylpentanoyl)piperazin-2-one
8-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
4-(5-methyl-1,2,4-oxadiazol-3-yl)-N-[3-(pyridin-3-yl)phenyl]piperidine-1-carboxamide
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-[1-(4-oxopentanoyl)piperidin-4-yl]imidazolidine-2,4-dione
(2E)-1-[4-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
(3aS,7aR)-5-methyl-2-(5-phenylpentanoyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
7-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(diphenylmethyl)-N-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(1-benzothiophen-2-ylmethyl)-1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(3-methyl-2-oxopyrrolidin-1-yl)acetamide
5-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-3-[(4-fluorophenyl)methyl]-5-methylimidazolidine-2,4-dione
(1S,5R)-6-benzyl-3-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(pentan-3-yl)amine
N-(furan-2-ylmethyl)-9-methoxy-7-oxo-3-{[4-(propan-2-yl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(5-{[cycloheptyl(pyridin-3-ylmethyl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
(3aS,6aR)-5-(4,6-dimethylpyrimidin-2-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-4-(piperidin-3-yl)benzamide
2-(2-methyl-1,3-thiazole-4-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
6-methyl-2-{[2-({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}amino)ethyl]amino}-3,4-dihydropyrimidin-4-one
3-{1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-3-carbonyl}pyridine
3-(1-benzofuran-2-ylmethyl)-9-methoxy-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-(1-methylcyclopropanecarbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3R,4S)-4-(4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1,4-diazepan-1-yl)oxolan-3-ol
N-cyclobutyl-3-{[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]sulfamoyl}benzamide
3-methyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-{[benzyl(cyclopentyl)carbamoyl]amino}-N,N,2-trimethylbenzamide
2-cyclopropyl-9-[3-(2,4-difluorophenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclohexyl-3-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}-N-methylpyridin-2-amine
1-[2-methoxy-5-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-(3-fluoro-4-methoxyphenyl)-6-(pyrrolidin-1-yl)pyridazine
N-[(3R,4S)-4-cyclopropyl-1-[2-(3-methoxyphenoxy)ethyl]pyrrolidin-3-yl]methanesulfonamide
4-(2,3-difluoro-4-methoxybenzoyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-amino-1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetamide
2-amino-N-[3-(pyridin-3-yl)propyl]-4-(trifluoromethyl)pyrimidine-5-carboxamide
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(4-methylpiperazin-1-yl)propan-1-one
{3-[(2-fluorophenyl)methyl]-1-[(8-fluoroquinolin-2-yl)methyl]piperidin-3-yl}methanol
2-ethoxy-6-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}phenol
4-(1-benzofuran-5-ylmethyl)-1-(3-methoxyphenyl)piperazin-2-one
1-{1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]azetidin-3-yl}-2-methylpiperidine
[(1R,3S,3aS,6aR)-5-methyl-1-(2-methylpropyl)-3-[2-(1H-pyrazol-1-ylmethyl)phenyl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
1-[2-(dimethylamino)-4-{[(5-methylpyrazin-2-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]acetamide
N3-cyclooctyl-N5-cyclopentyl-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-4-(thiophen-2-yl)butanamide
5-methyl-N,N-bis(prop-2-en-1-yl)-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-(2-methylprop-2-en-1-yl)-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide