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6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1,4-diazepan-2-one
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-(1-methyl-1H-pyrazole-5-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(1-cyclopentanecarbonylpiperidine-4-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
(2,3-dihydro-1-benzofuran-5-ylmethyl)({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl})amine
2-(oxolan-2-ylmethoxy)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}amine
2-(1-{2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-2-yl)ethan-1-ol
3-(2H-1,3-benzodioxol-5-yl)-5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
N-methyl-N-(quinolin-6-ylmethyl)-3-(trimethyl-1H-pyrazol-1-yl)propanamide
1-benzyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-{[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperazin-1-yl]methyl}benzoic acid
4-(2-cyclopropyl-1,3-benzoxazol-5-yl)benzamide
N-cyclopropyl-3-{1-[2-(naphthalen-1-yl)acetyl]piperidin-4-yl}propanamide
2-ethyl-8-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2,8-diazaspiro[4.5]decan-3-one
3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-methyl-2-(morpholin-4-yl)propyl]acetamide
1-ethyl-8-{[4-(furan-2-yl)phenyl]methyl}-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-N-methyl-1-[(2E)-2-methylbut-2-en-1-yl]-4-[2-(pyridin-4-ylsulfanyl)acetamido]pyrrolidine-2-carboxamide
1-(1,2-oxazole-3-carbonyl)-4-phenyl-1,4-diazepane
N,3,5-trimethyl-N-[1-(pyridin-3-yl)ethyl]-1,2-oxazole-4-carboxamide
3-(3,4-dimethoxybenzoyl)-1-(2,3,4-trimethoxybenzoyl)piperidine
8-(3-hydroxy-2-methylbenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl (2R)-2-({2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)propanoate
3-acetamido-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
2-methyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-(thiophen-2-ylformamido)propanamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(1,3-thiazol-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-ethoxyphenyl)ethan-1-one
N-[(3R,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-(3,4-dimethylphenyl)propanamide
1-(3-fluorophenyl)-3-(furan-2-yl)-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
8-(6-methoxyhexanoyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(furan-3-carbonyl)piperidine-4-carboxamide
(1R,5S,6R)-3-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
1-{[1-(6-{[2-(dimethylamino)ethyl]amino}pyridine-3-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
methyl 3-[(2-ethylbutanamido)methyl]-5-[2-(thiophen-3-yl)acetamido]benzoate
3-{[4-(3-chlorophenyl)-5-{[methyl(quinoxalin-5-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
1-(2,2-dimethylpropyl)-3-({[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-3-hydroxypiperidin-2-one
2-{[(4aS,7aR)-6,6-dioxo-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
[(3R,4R)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-(2-methoxyethyl)-8-(4-propylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(4-methylphenoxy)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-methyl-N-(quinolin-5-ylmethyl)-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
2-[2-(phenylsulfanyl)ethyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
N-[2-(4-methylpiperidin-1-yl)ethyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxamide
3-[5-(2,3,6-trimethylphenoxymethyl)-1,2,4-oxadiazol-3-yl]pyridazine
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[4-(8-methoxy-2-methylquinolin-5-yl)-1H-pyrazol-1-yl]acetamide
5-(1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-1H-imidazol-2-yl)-2,1,3-benzoxadiazole
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
methyl (2S)-1-[1-(4-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)piperidin-4-yl]pyrrolidine-2-carboxylate
2-(1-propylpiperidin-4-yl)-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethan-1-one