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3-(1H-1,3-benzodiazol-2-yl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
1-[(4-methoxyphenyl)methyl]-N,N-bis(prop-2-en-1-yl)-1H-1,2,3-triazole-4-carboxamide
2-(pyrrolidin-1-yl)-5-{1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-2-yl}pyrimidine
2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[(4-methylphenyl)methyl]acetamide
4-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-4-(morpholin-4-yl)butan-1-one
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N,N-bis(prop-2-en-1-yl)benzamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
3-(4-fluorophenyl)-4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperazin-2-one
1-(1-cyclopropylethyl)-5-(2-ethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]propanamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N,N-diethyl-4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepan-6-ol
(2S)-2-acetamido-3-[1-(3-methylpyridin-2-yl)-1H-imidazol-4-yl]propanoic acid
5-oxo-1-phenyl-N-[1-(pyridin-2-yl)propan-2-yl]-2,5-dihydro-1H-pyrazole-3-carboxamide
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-(pyrazine-2-carbonyl)piperidin-4-amine
1-(4,6-dimethylquinazolin-2-yl)-N-ethylpiperidine-4-carboxamide
N-ethyl-8-methoxy-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-(oxan-4-yl)piperidin-3-amine
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[1-(thiophen-3-yl)propan-2-yl]acetamide
methyl 5-{[(4-ethoxyphenyl)methyl]amino}-1-(2-methoxyethyl)-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3R,4S)-4-{[(2,6-dichloro-3-hydroxyphenyl)methyl](methyl)amino}oxolan-3-ol
4-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1-(4-methylphenyl)piperazin-2-one
6-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-sulfonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-4-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetyl)-1,4-diazepan-2-one
3-({1-[(3-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
1-[3-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)propyl]-1H-imidazole
4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazine-1-sulfonamide
2-[4-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-1-(2,2-dimethylpropyl)piperazin-2-yl]ethan-1-ol
4-({1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-2-yl}methyl)morpholine
3-({5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}formamido)-N-(2-methylphenyl)propanamide
1-[2-hydroxy-3-(4-methoxy-2-{[methyl(prop-2-en-1-yl)amino]methyl}phenoxy)propyl]piperidin-4-ol
1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
2-(4-{[2-hydroxy-3-(pyrrolidin-1-yl)propyl]amino}-6-methylpyrimidin-2-yl)phenol
9-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(1H-imidazol-2-ylmethyl)(methyl)[(3-{[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
(3S,4S)-4-(dimethylamino)-1-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-ol
N-{[2-(benzyloxy)phenyl]methyl}-1-(carbamoylmethyl)piperidine-4-carboxamide
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-4-(thian-4-yl)piperazine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}urea
N-(3-hydroxy-2,2-dimethylpropyl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-[benzyl(methyl)amino]-N-(1,4-dioxan-2-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
3-methoxy-2,2-dimethyl-1-(3-phenylpiperazin-1-yl)propan-1-one
2-chloro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
3-({4-[3-(2-phenylethyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
methyl 6-[(4-phenylpiperidin-1-yl)methyl]-3-propanamidothieno[2,3-b]pyridine-2-carboxylate