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N-cyclopropyl-5-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-{[4-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazole
4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole
6-chloro-8-methyl-3-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
N-[2-(diethylamino)ethyl]-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carboxamide
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-[1-(thiophen-3-yl)propan-2-yl]acetamide
8-fluoro-N-(furan-3-ylmethyl)-N-methylquinoline-2-carboxamide
2-methyl-N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}benzene-1-sulfonamide
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-[1-(2-methylquinoline-4-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1,3-dimethyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(1,3-benzothiazol-2-yl)-N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]pyrrolidine-1-carboxamide
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(4-methylphenyl)propanamide
{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2,3-dimethoxy-N-{[7-(methylsulfanyl)-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
1-{1-[2-(2-chlorophenoxy)acetyl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
3-phenyl-N-(1-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
4-{[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}benzoic acid
N-(3-fluorophenyl)-6-(9-methyl-9H-carbazole-3-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
{3-benzyl-1-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
4-({1-[3-(3-chlorophenyl)phenyl]piperidin-4-yl}amino)butan-1-ol
1-(2-methoxyphenyl)-3-(1-{1-[3-(1-methylcyclopropyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-cyclopropyl-1-[1-(furan-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(3aS,6aS)-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)-5-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[2-(3-methoxyphenyl)ethyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-3-phenoxypropanamide
(1R,9aR)-1-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxymethyl]-octahydro-1H-quinolizine
N-{[1-(dimethylamino)cyclohexyl]methyl}-4-(3-hydroxy-3-methylbutyl)benzamide
N-(oxolan-2-ylmethyl)-3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
1-({1-[3-(propan-2-yloxy)benzoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
(2S,4R)-4-{[(4-fluorophenyl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-cyclopropyl-3-[1-(5-fluoro-1H-indole-2-carbonyl)piperidin-4-yl]propanamide
2-cyano-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}benzamide
methyl 2-[3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamido]acetate
9-(cyclopropylmethyl)-1-methyl-4-(5-methyl-1,3-oxazole-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)-N-methyl-N-[2-(pyridin-2-yl)ethyl]acetamide
5-[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]-4-methyl-1,3-thiazol-2-amine
1-benzyl-8-[(4-methoxy-3-methylphenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-2-amino-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-imidazol-4-yl)propan-1-one
8-methoxy-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-yl]acetamide
2-methyl-6-[(3-propylmorpholin-4-yl)methyl]phenol
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-2,5-dimethoxy-N-(pyridin-3-ylmethyl)benzene-1-sulfonamide
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(5-fluoro-2-methylphenyl)ethan-1-one
8-[3-(4-methylphenyl)propanoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(2-methylpropyl)-N-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
propyl 4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide