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2-(1H-1,3-benzodiazol-1-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]propanamide
(2S,4R)-4-amino-1-[4-(1H-indol-3-yl)butanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[(5-ethylfuran-2-yl)methyl]-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[2-chloro-4-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]acetamide
1-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(2-methyl-1-benzofuran-5-yl)urea
N-cyclopentyl-3-{[(4-methoxy-3-methylphenyl)methyl]amino}-5-(phenylsulfamoyl)benzamide
N-(pyridin-2-ylmethyl)-3-{[1-(thiophen-3-ylmethyl)piperidin-4-yl]oxy}benzamide
3,3-dimethyl-1-[(3S,4R)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-(propan-2-yl)pyrrolidin-3-yl]urea
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-methylpropanamide
1-[(4aR,8aR)-7-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
2-(5-acetylthiophen-3-yl)-N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]acetamide
N-{[1-(isoquinolin-5-ylmethyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
2-amino-6-cyclopropyl-4-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
N-[2-(dimethylamino)ethyl]-5-(pyrazine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(2-methoxy-2-methylpropyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-{[1-(2-methoxy-4-methylbenzenesulfonyl)piperidin-2-yl]methyl}morpholine
5-[(4-chlorophenyl)methyl]-5-{3-[3-(3-methylphenyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-methyl-1'-(5-methyl-1H-indazole-3-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]amine
N-(2,3-dimethylphenyl)-2-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]amino}acetamide
2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(2S,4R)-4-(4-chlorobenzamido)-1-(3-methylbut-2-en-1-yl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-(hydroxymethyl)-1-[3-(1H-imidazol-2-yl)benzoyl]azepan-4-ol
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-[1-(thiophen-2-yl)propyl]piperidine-4-carboxamide
1-[1'-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
6-methoxy-3-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1-benzofuran-2-carboxamide
2-(adamantan-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-3-methylbenzamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-(1H-pyrazol-4-yl)butanamide
2-(2-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
1-[(5-chlorofuran-2-yl)methyl]-4-(4-fluorophenyl)-1,4-diazepane
N-[2-(cyclohexylsulfanyl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[(2E)-2-methylbut-2-en-1-yl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
(1s,4s)-N1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]cyclohexane-1,4-diamine
5-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[3-(ethoxymethyl)-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
1-(3-methoxybenzoyl)-4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
2-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-6-methyl-4H-pyran-4-one
4-(pyridin-2-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
5-({5-[4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazol-5-yl]furan-2-yl}sulfanyl)-1H-1,2,4-triazole
2-[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
1-[4-(3-methoxyphenoxy)phenyl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea
N-(2,6-dimethoxypyridin-3-yl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
2-(5-chlorothiophene-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-ethyl-1-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
1-(1-benzothiophen-2-yl)-2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethan-1-ol
4-[(3-{3-cyclopropyl-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]morpholine
2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-imidazole
(3aR,6aR)-2-(pyridine-3-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid