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2-(cyclopropylmethyl)-8-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
1-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-(pyridin-4-yl)piperazine
3-[1-ethyl-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]-4-methylbenzene-1-sulfonamide
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
3-amino-1-[(1-phenyl-1H-pyrazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
3-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]ethan-1-one
2-(2-hydroxyethyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-1-carboxamide
5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole
1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-(3-chlorophenyl)-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
2-(adamantan-1-yl)-4-hydroxy-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidine-5-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[(dimethylamino)methyl]-1,3-thiazole-4-carboxamide
4-(dimethylsulfamoyl)-N-[3-(1,3-oxazol-5-yl)phenyl]piperazine-1-carboxamide
2-(2,4-difluorophenyl)-8-methoxy-5-[(2-methyl-1H-imidazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}-1H-indole
N-[(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-4-yl)methyl]acetamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
6-methyl-3-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-ethyl-N-methyl-3-({2-[(pyridin-3-yl)amino]ethyl}sulfamoyl)benzamide
N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
6-methyl-5-(morpholine-4-carbonyl)-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,3,4-tetrahydropyrimidin-2-one
2-ethyl-1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
7-butoxy-4-(3-fluoropyridin-4-yl)-1,2,3,4-tetrahydroquinolin-2-one
10-methoxy-5-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-[2-(2,4-difluorophenyl)-1-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
2-ethyl-4-phenyl-9-(pyrrolidine-1-carbonyl)-2,9-diazaspiro[5.5]undecane
N-[2-(1H-imidazol-4-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(2R,3R,6R)-5-(5-methyl-1,2-oxazole-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}-1-[3-(sulfamoylmethyl)phenyl]urea
N-[(3R,4S)-1-(1-aminocyclopropanecarbonyl)-4-cyclopropylpyrrolidin-3-yl]-6-methylpyrimidin-4-amine
(3ar,6ar)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-4-yl}propanamide
2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)amino}-1-(4-hydroxyphenyl)ethan-1-one
4-methyl-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,4-diazepan-5-one
2-fluoro-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzene-1-sulfonamide
[(2-butyl-1H-imidazol-4-yl)methyl]({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl})(2-methoxyethyl)amine
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methoxypyridine-3-carboxamide
2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
4-[1-(2,6-dimethoxypyridin-3-yl)-1H-imidazol-2-yl]-2-ethylpyrimidine
1-(4,6-dimethylquinazolin-2-yl)-N-(3-hydroxyadamantan-1-yl)piperidine-4-carboxamide
3-[(2-fluorophenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-cyclopropyl-N-(1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
(3S,4S)-4-cyclopropyl-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidine-3-carboxylic acid
N-(3-hydroxypropyl)-1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
3-[(2,4-dimethoxyphenyl)methyl]-9-methoxy-10-(4-methylpiperazine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(propan-2-ylsulfanyl)acetamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}amine
3-(1H-1,2,3-benzotriazol-1-yl)-1-(4-cyclopentyl-1,4-diazepan-1-yl)propan-1-one
6-[3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carbonyl]-2-methyl-2,3,4,5-tetrahydropyridazin-3-one