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N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]cyclopropanesulfonamide
2-[(3-fluorophenyl)methyl]-4-[4-(pent-4-enoyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-(1-methyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(5-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}furan-2-yl)benzonitrile
6-(2-butoxy-4-fluorophenyl)-5-chloro-2-methylpyrimidin-4-ol
1-methyl-N-({1-[(2E)-2-methylpent-2-en-1-yl]pyrrolidin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[5-({[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
(3S)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-N,N-dimethylazepan-3-amine
1-[(3R)-3-cyclopropyl-3-hydroxy-4,4-dimethylpyrrolidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
2-{3-cyclopentyl-5-[4-(1H-pyrazol-3-yl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
6-(dimethyl-1,3-thiazole-5-carbonyl)-3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(dimethylamino)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-(2-methylphenyl)acetamide
(benzylsulfamoyl)[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]amine
2-methyl-1-(2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}-2-oxoethyl)-1H-indole-3-carbonitrile
(1S,3R)-3-amino-N-{2-[ethyl(3-methylphenyl)amino]ethyl}cyclopentane-1-carboxamide
3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-[3-(propan-2-yloxy)propyl]propanamide
7-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[3-(1H-pyrazol-1-yl)phenyl]-1-(pyridine-2-carbonyl)pyrrolidine-2-carboxamide
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-3-(2-methoxyphenyl)-N-[(3S)-2-oxoazepan-3-yl]propanamide
{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
1-{5-[5-(5-cyclopropyl-1,2-oxazol-3-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}-2-methylpropan-1-one
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-4-yl)propan-1-one
4-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1-phenylpiperazin-2-one
1-[2-(methylsulfanyl)benzoyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
2-[4-(7-chloroquinolin-4-yl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
[2-(azepan-1-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(propan-2-yl)amine
N,N-diethyl-1-[1-(4-fluorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-(4-methoxybutyl)-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine
1-cyclopentyl-4-(2-methoxypyridine-4-carbonyl)-1,4-diazepane
N-{5-[1-(2-hydroxyethyl)-1H-imidazol-2-yl]pyrimidin-2-yl}benzenesulfonamide
{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-cyclopentyl-3-{2-[4-(1-hydroxypropyl)piperidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
[9-(pyridin-4-ylmethyl)-3-(thiophene-3-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
N-(1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(2-hydroxyphenyl)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyrrolidine-2-carboxamide
9-(2-aminopyridine-4-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-6-(2,1,3-benzothiadiazol-5-ylmethyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
[(3-methyl-1H-pyrazol-5-yl)methyl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine
5-cyclobutyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1,3,4-oxadiazol-2-amine
2-[1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidin-2-yl]pyridine
2-[5-(3-fluoro-2-methoxyphenyl)-3-phenyl-1H-1,2,4-triazol-1-yl]pyridine
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
2-{[2-(dimethylamino)ethyl](methyl)amino}-N-[(4-methoxyphenyl)methyl]-6-[4-(methylsulfanyl)phenyl]pyridine-3-carboxamide
1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
(4aS,8aR)-6-[(2-phenyl-1,3-thiazol-4-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
(2S)-2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-3-methylbutanamide
{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine