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N-(butan-2-yl)-3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
5-chloro-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-3-phenyl-1H-indole
4-methyl-N-(3-methyl-4-pentanamidophenyl)-3-(2-oxoimidazolidin-1-yl)benzamide
4-(6-chloro-2H-1,3-benzodioxol-5-yl)-5,6,7-trimethoxy-1,2,3,4-tetrahydroquinolin-2-one
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
4-[1-(5-chloro-2-fluorobenzoyl)piperidin-4-yl]-5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidine
1-[2-(dimethylamino)-4-{methyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(2E)-1-(4-{1-[(2-methoxyethyl)(pyridin-2-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-3-phenylprop-2-en-1-one
3-({2-ethyl-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-1λ6-thiolane-1,1-dione
3-[(4-fluorophenyl)methyl]-5-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
3-{[methyl({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl})amino]methyl}phenol
3-[3-(dimethylamino)propyl]-5-[(4-fluorophenyl)methyl]-5-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
(3S,5R,9R)-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1H-1,2,3-triazole-5-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-{2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]ethyl}-1,3-oxazolidin-2-one
1-(4-chlorophenyl)-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropane-1-carboxamide
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-[1-(pyrazin-2-yl)propan-2-yl]propanamide
N4-cyclopropyl-7-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]propan-1-one
2-ethyl-4-methyl-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1,3-thiazole-5-carboxamide
5-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
N-benzyl-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-(pyridin-3-ylmethyl)-3-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]propanamide
N-(2H-1,3-benzodioxol-5-yl)-4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carboxamide
N-(4-{[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]methyl}phenyl)acetamide
1-(2-chlorophenyl)-4-[3-(3-methoxyphenyl)propanoyl]piperazin-2-one
2-methoxy-N-(7-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1-(2-phenylethyl)-1H-1,3-benzodiazol-5-yl)acetamide
1-(4-{2-[2-(2-methoxyphenyl)ethyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-({7-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(4-phenylbutyl)-2-(propan-2-yl)pyrimidine-5-carboxamide
3-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxylic acid
1-[(3-chloro-4-ethoxyphenyl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-[({[4-(3-chlorophenyl)-5-[(3-hydroxypropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-2-ethoxyphenol
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
7-(cyclobutylmethyl)-2-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,7-diazaspiro[4.5]decane
(2S,4R)-4-amino-N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)pyrrolidine-2-carboxamide
2-[4-(benzyloxy)piperidin-1-yl]-5-(1H-imidazol-1-ylmethyl)pyridine
2-[(4-fluorophenyl)methyl]-4-(1-methyl-1H-pyrazole-5-carbonyl)morpholine
4-{1-benzyl-5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-6-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
2-{4-[(3-methylquinoxalin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
8-[4-(1H-imidazol-1-yl)butanoyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-oxo-4-phenylbutanamide
N-(1-{1-[2-(2-chlorophenoxy)acetyl]piperidin-4-yl}-2-(2,4-difluorophenyl)ethyl)-N-methylpropanamide
7-chloro-N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]quinoxalin-2-amine
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
2-oxo-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,2-dihydroquinazoline-4-carboxamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide