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1-[3-(1,2-oxazinan-2-yl)propanoyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
1-{3-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[2-oxo-2-(piperidin-1-yl)ethyl]-4-(pyridin-2-ylmethyl)piperazin-2-one
2-{1-cyclopentyl-4-[(3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-1-(pyridin-2-ylmethyl)piperidin-4-amine
N-[2-(2-methoxyphenyl)ethyl]-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[2-(pyridin-3-yl)ethyl]pyrimidin-2-amine
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
3-[3-(4-chlorobenzoyl)piperidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
N-(1-{7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
N-[(3S,4R)-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-(4-carbamoylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-{4-[3-(2-methylpropoxy)phenyl]-1H-pyrazol-1-yl}propanamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
4-phenyl-1-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
(4aR,7aS)-1-acetyl-4-(5-methylpyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S)-1-{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-(1H-imidazol-2-yl)benzamide
N-methyl-3-(3-methylpiperidin-1-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
6-{1-[4-(pyridin-3-yl)pyrimidin-2-yl]piperidin-3-yl}pyrimidin-4-ol
5-chloro-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
(3aS,6aR)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
N-({7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
4-[2-(1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-2-yl)ethyl]morpholine
6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(methylsulfanyl)pyrimidin-4-amine
ethyl 5-({[2-(propan-2-yl)-1,3-benzoxazol-5-yl]formamido}methyl)furan-2-carboxylate
4-[6-(propan-2-yl)-1H-indole-2-carbonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
methyl (1R,3S,3aR,6aS)-3-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[(2R,3R)-2-hydroxy-1'-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
2-{4-[(1R,9aR)-octahydro-1H-quinolizine-1-carbonyl]piperazin-1-yl}benzonitrile
7-(4-fluoro-2-methylbenzoyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3,5-dimethoxy-N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)benzamide
1-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[3-(4-methyl-1,3-thiazol-2-yl)propyl]urea
2-(4-fluorophenyl)-1-[4-(pyrrolidin-1-yl)benzoyl]pyrrolidine
ethyl 5-{spiro[2.4]heptane-1-carbonyl}-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1R,5R)-3-methanesulfonyl-6-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
4-methyl-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pentane-1,2-dione
methyl 4-oxo-4-{4-[2-(phenylcarbamoyl)ethyl]piperidin-1-yl}butanoate
5-{3-[4-(2,3-dimethylphenyl)piperazin-1-yl]-3-oxopropyl}-5-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-2-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-ol
4-{3-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
(1R,5S)-3-[2-(1H-indol-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(3R,4S)-1-(3-chloro-4-fluorobenzoyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
1-(furan-2-carbonyl)-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazine
1-(5-methylpyridine-3-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1-methylcyclopropyl)propanamide