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4-benzyl-1-(5-methanesulfonyl-2-methylpyrimidin-4-yl)piperidin-4-ol
(4aR,7aS)-N-(2,1,3-benzothiadiazol-4-yl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
6-(morpholine-4-carbonyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrazin-2-amine
2-(3,5-difluorophenyl)-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
N-[3-(pyridin-3-yloxy)propyl]-3-azaspiro[5.5]undecan-9-amine
2-tert-butyl-7,7-dimethyl-N-(pyridin-2-ylmethyl)-5,6,7,8-tetrahydroquinazolin-5-amine
4-[4-(piperidine-1-carbonyl)piperidin-1-yl]-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-(cyclopropylmethyl)-5-[1-(2,5-difluorobenzoyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
N-{[7-(1H-1,3-benzodiazole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
2-(2-methoxy-5-methylbenzenesulfonyl)-2,8-diazaspiro[4.5]decane
{1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
2-{4-[(3,4-dimethoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
methyl 3-acetamido-1-(3-methylbutyl)-5-[(6-methylhept-5-en-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2,1,3-benzoxadiazol-5-ylmethyl)({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
ethyl 2-[1-(5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazol-3-yl)-N-methylformamido]acetate
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-methyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
N-methyl-1-(3-phenylpropyl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-amine
7-(propan-2-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-benzyl-2-cyclobutaneamido-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
3-[6-amino-4-(2-butyl-1H-imidazol-4-yl)-5-cyanopyridin-2-yl]-1H-pyrazole-5-carboxylic acid
5-{4-azatricyclo[4.3.1.13,8]undecan-4-yl}-1-(3-methylbutyl)azepan-2-one
N-methyl-1-(2-methyl-6-propylpyrimidin-4-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)piperidin-4-amine
N-(1H-1,3-benzodiazol-2-ylmethyl)-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(3-methoxyphenyl)-1-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
6-(trifluoromethyl)-3-[2-(trifluoromethyl)morpholine-4-carbonyl]pyridin-2-ol
N-methyl-5-(oxolan-2-yl)-N-(thiophen-3-ylmethyl)thiophene-2-carboxamide
2-methyl-5-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-3,4-dihydropyrimidin-4-one
[(3R,4R)-1-[4-(5-methylfuran-2-yl)benzoyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-(prop-2-en-1-yl)-9-[4-(trifluoromethyl)pyrimidin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[2-(pyridin-2-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
ethyl 1-[5-acetamido-2-ethyl-1-(pyridin-3-ylmethyl)-1H-1,3-benzodiazole-7-carbonyl]piperidine-2-carboxylate
2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-N-(1,2-oxazol-3-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[(3R,4S)-3-(6-methyl-4-oxo-1,4-dihydropyridine-3-amido)-4-(propan-2-yl)pyrrolidin-1-yl]butanoic acid
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]amine
N-[4-(5-methyl-4-{[3-(thiophen-2-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-3-carboxamide
5-{[methyl({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl})amino]methyl}pyrimidin-2-amine
2-(2,3-difluorophenoxymethyl)-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
3-{1-[5-(propan-2-yl)-1,2-oxazol-3-yl]-N-(pyridin-3-ylmethyl)formamido}propanoic acid
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-[(2R,3R)-1'-(3,5-difluorobenzoyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
5-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
N-[2-(2-methoxyphenyl)ethyl]-6-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-6-azaspiro[2.5]octane-1-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-[3-(1H-indol-1-yl)propyl]-1,1-dioxo-1λ6-thiolane-3-carboxamide
3,4-dimethoxy-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
5-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]quinoxaline