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(2S,4S)-1-benzyl-N-ethyl-4-[(1-ethylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
11-methyl-4-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[6-hydroxy-4-(2-methylpropyl)-1,4-diazepan-1-yl]-1,3-thiazole-4-carboxamide
1-(2-methoxyethyl)-3-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(6-hydroxypyrimidin-4-yl)methyl]acetamide
1-{[1-(1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]methyl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
N-[(2R,3R)-1'-[(4-chlorophenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanoyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-(1H-imidazol-2-yl)piperidine
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-[2-(furan-2-yl)ethyl]pyridin-2-amine
(3S,5R)-N-(6-methylpyridin-3-yl)-5-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)piperidine-3-carboxamide
N-(3-methoxypropyl)-5-methyl-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-{2-[2-(1-benzothiophen-2-yl)-1H-imidazol-1-yl]ethyl}acetamide
methyl (2S,4S,5R)-4-(cyclobutylcarbamoyl)-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylate
N-(5-aminopentyl)-1-benzofuran-3-carboxamide
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
1-(cyclopropylmethyl)-5-[2-(3,4-difluorophenyl)acetyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-(isoquinolin-5-yl)urea
1-({4-[(2,5-dimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-4-ol
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-N-(4-methylphenyl)piperidine-1-carboxamide
5-cyclopropanecarbonyl-1'-(oxan-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(3-cyclopropyl-1H-pyrazol-5-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
4-(1H-imidazol-1-ylmethyl)-5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazole
[(3R,4R)-1-(4-chloro-2-fluorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
9-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
5-(propan-2-yl)-N-[2-(pyridin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N2,N2-dimethyl-N5-[(5-methylthiophen-2-yl)methyl]-5,6,7,8-tetrahydroquinazoline-2,5-diamine
N-[(3S,4R)-4-(propan-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]pyrrolidin-3-yl]acetamide
N-(1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
5-{2-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]ethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(2-methoxyphenyl)methyl]methylamine
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazole
1-[1-(3-fluorobenzoyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
1-(2-methoxyethyl)-N3-(1-methoxypropan-2-yl)-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
(5S,9aS,9bS)-5-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(2-chloro-6-fluorophenyl)methyl]-3-methyl-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-yl}-1H-1,2,4-triazole
5-(2,3-dimethoxybenzoyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-[2-(dimethylamino)ethyl]-6-oxo-N-[4-(pyridin-2-yl)butyl]piperidine-3-carboxamide
2-(2-hydroxypropyl)-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
(1-{[6-(2,3-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2,5-dihydro-1H-pyrrol-2-yl)methanol
4-(dimethylamino)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-3-(4-ethylphenyl)-1H-pyrazole
5-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2,4-dimethyl-N-{1-[4-(morpholine-4-carbonyl)phenyl]-1H-pyrazol-4-yl}benzamide
5-ethyl-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]pyrazolo[1,5-a]pyrimidin-7-amine
[(2-fluorophenyl)methyl](2-methoxyethyl){[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}amine
N-[3-(3,4-dimethylphenoxy)propyl]-N-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide