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3-(2-fluoro-4-methoxyphenyl)-1-phenyl-4-(pyrrolidin-1-ylmethyl)-1H-pyrazole
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}propan-1-one
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-[2-(pyrazin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(propan-2-yl)propanamide
2-(4-{[3-(2-methylphenyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-({5-[1-(furan-2-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
(3R,4S)-4-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1,4-diazepan-1-yl]oxolan-3-ol
2-butyl-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-benzoxazole-5-carboxamide
2-[2-({methyl[(1,2,2-trimethylpyrrolidin-3-yl)methyl]amino}methyl)phenoxy]acetic acid
2-(2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-[(2-chlorophenyl)methyl]-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
2,6-dimethyl-5-{2-oxo-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
3-methyl-8-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
2-(cyclopropylmethyl)-7-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-fluoro-2-(2-methoxypyridin-3-yl)phenol
4-({methyl[1-(methylcarbamoyl)propan-2-yl]amino}methyl)-N-phenylbenzamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl]urea
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-indol-1-yl)ethyl]acetamide
(2S,4S)-4-amino-1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-N,N-diethylpyrrolidine-2-carboxamide
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-3-carbonyl]piperidine
N-{[7-(2,3-dimethoxybenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
7-fluoro-2-methyl-3-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-indol-3-yl)ethyl]acetamide
ethyl 1-[4-(dimethylamino)benzoyl]-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
{[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl}[(3,4,5-trimethoxyphenyl)methyl]amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetamide
N-cyclohexyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
2-({methyl[2-(oxan-2-yl)ethyl]amino}methyl)benzoic acid
1-(azepan-1-yl)-3-[4-chloro-2-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-{1-methyl-5-[4-(1H-pyrazol-1-yl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1-[(1R,2S)-2-phenylcyclopropyl]-1H-imidazole
7-(2,1,3-benzothiadiazole-4-sulfonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2S,4S,5R)-4-[(2,2-difluoroethyl)carbamoyl]-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
N-(1-methylpiperidin-4-yl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-(furan-2-yl)-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]azepane
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,4,6-trimethoxyphenyl)methyl]piperidine
N,N-diethyl-2-[1-(2-methoxyethyl)-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
3-{5-[3-(methylsulfanyl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
2-(2-chloro-6-methoxyphenyl)-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]acetic acid
1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[(4-methyl-1,3-thiazol-2-yl)methyl]urea
1-[2-(4-methoxyphenyl)ethyl]-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-2-one
1-[3-(furan-2-yl)phenyl]-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-amine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(2-phenyl-1H-imidazol-1-yl)acetamide
(2-methoxyethyl)({8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl})(oxolan-2-ylmethyl)amine