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2-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(ethyl)amino)ethan-1-ol
1-(carbamoylmethyl)-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
[1-(quinolin-4-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
9-methyl-3-(pyridin-4-ylmethyl)-3,9-diazaspiro[5.6]dodecan-10-one
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyridine-3-sulfonamide
1-[5-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2-methylphenyl]imidazolidin-2-one
1-{[1-(5-phenyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
4-(3-hydroxy-3-methylbutyl)-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-(5-fluoro-2-methoxyphenyl)-2-{4-[2-(2-hydroxyethoxy)ethyl]piperazin-1-yl}acetic acid
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-[1-hydroxy-2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]phenol
2,6-dimethyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]quinoline-3-carboxamide
ethyl 2-{1-[2-(2-methoxyethyl)-1,3-benzoxazole-6-carbonyl]piperidin-2-yl}acetate
N-methyl-N-[(4-methylphenyl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpiperidin-4-yl)methyl]amine
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
7-methyl-4-(pyrrolidin-3-ylmethyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-(furan-3-ylmethyl)-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
4-(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-2-oxopiperazin-1-yl)benzonitrile
1-cyclohexyl-4-[2-(1-methyl-3-oxopiperazin-2-yl)acetyl]piperazin-2-one
4,6-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carboxamide
2-amino-4-[2,5-dimethoxy-4-(methylsulfanyl)phenyl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methyl-1,3-oxazole-4-carboxamide
N-(3-methoxyphenyl)-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propanamide
2-methyl-4-(4-{[(1R,5S,6S)-6-(4-methylpiperazine-1-carbonyl)-3-azabicyclo[3.1.0]hexan-3-yl]methyl}phenyl)but-3-yn-2-ol
1-(3-propyl-1H-pyrazole-4-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
1-(3-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2,2-dimethylbutan-1-one
6-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[(2-fluorophenyl)formamido]-N-methylpropanamide
N-[(3-methyl-7-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-2-sulfonamide
(1S,2R)-N1-[2-(4-methoxyphenyl)propan-2-yl]-N2-propylcyclohexane-1,2-dicarboxamide
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-(2-phenylpropyl)-1H-1,2,3-triazole
4-chloro-1,5-dimethyl-N-(4-phenylbutyl)-1H-pyrazole-3-carboxamide
2-{1-[(3,4-dimethoxypyridin-2-yl)methyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpyrrolidine-2-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclopropanesulfonamide
(3R,4R)-4-(azepan-1-yl)-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-ol
3-(1-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1H-imidazol-2-yl)pyridin-2-amine
N-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-2-phenylpiperidine-1-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-[1-cyclohexyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
2-(2,3-dimethylphenoxy)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(2-chlorophenyl)-3-phenyl-N-[(1s,4s)-4-aminocyclohexyl]propanamide
3-(methylsulfanyl)-1-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
ethyl 1-benzyl-5-[(5-acetamidothiophen-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-[(2,3-difluorophenyl)methyl]-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
N-{1-[1-(2-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
N-(2-phenylethyl)-6-(2-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[(2R,4R,6S)-2-phenyl-6-[4-(pyridin-2-yl)phenyl]oxan-4-yl]acetamide