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1-[(3,4-dimethylphenyl)methyl]-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazin-2-one
N-({7-[2-(cyclohex-1-en-1-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-6-(dimethylamino)pyridine-3-carboxamide
7-acetamido-1-[2-(pyridin-2-yl)ethyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-1,3-benzodiazole-5-carboxamide
4-(hydroxymethyl)-1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}azepan-4-ol
9-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-tert-butyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
(4S,6R)-N-ethyl-6-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-2-sulfanylidene-1,3-diazinane-4-carboxamide
1-[2-(1H-imidazol-1-yl)ethyl]-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
1-(4-hydroxypiperidin-1-yl)-3-{5-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
7-(morpholine-4-sulfonyl)-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
3-[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
3-(2,5-difluorobenzoyl)-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
N-methyl-6-oxo-1-(3-phenylpropyl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethyl-2-oxoimidazolidine-4-carboxamide
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
1-{2-[(4-methoxyphenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
3-[5-(furan-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
6-{[methyl(thiophen-3-ylmethyl)amino]methyl}-2-oxo-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,2-dihydropyridine-3-carboxamide
N-(1-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2,1,3-benzoxadiazole-5-carboxamide
2-{1-[(5-methylfuran-2-yl)methyl]-4-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-cyclohexyl-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazine
(2E)-3-(3-fluorophenyl)-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}prop-2-enamide
6-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
(3S,5R)-1-benzoyl-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
3-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-methyl-2-phenyl-2-({2-phenylimidazo[1,2-a]pyridin-6-yl}formamido)acetamide
2-methyl-2-{2-[methyl(2-methylpropyl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}propanoic acid
5-{1-[(2,6-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
1-[(6-methoxypyridin-3-yl)methyl]-4-(oxan-4-yl)piperazine
1-[2-(dimethylamino)acetyl]-N-[4-(1H-indol-2-yl)phenyl]pyrrolidine-2-carboxamide
8-[(5-methylfuran-2-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-(5-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
N-tert-butyl-3-[2-(6-chloropyridin-3-yl)acetamido]-2-methylbenzamide
4-methyl-N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]pentanamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
(1R,5R)-N-(2-methoxyphenyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-cyclobutanecarbonyl-1'-(5-methyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-pyrazol-1-yl)butan-1-one
N-[2-(4-fluorophenyl)ethyl]-2-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]acetamide
4-({[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)amino}methyl)-1-cyclopentylpyrrolidin-2-one
1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(thiophen-2-yl)propan-1-one