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1-{5H,6H-benzo[h]quinazolin-2-yl}-N,5-dimethyl-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-4-carboxamide
7-(ethanesulfonyl)-N4-(1,2-oxazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-(3-chloro-4-fluorophenoxy)-1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[(2S,4R,6S)-2-ethyl-6-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]oxan-4-yl]acetamide
6-methyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylacetamide
1-(cyclopropanesulfonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-oxazepan-6-ol
5-{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
ethyl 1-(3-phenylpropyl)-5-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-amino-6-(2,4-dichlorophenyl)-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
(4aR,7aS)-1-methyl-4-(5-phenoxyfuran-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
1-(4-methylphenyl)-4-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}piperazin-2-one
(4aS,8aR)-6-[(4-chloro-3-fluorophenyl)methyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
N-(1H-indol-3-yl)-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-fluoro-N-[1-(4-methoxyphenyl)propyl]-5-sulfamoylbenzamide
5-methyl-N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-3-phenyl-1,2-oxazole-4-carboxamide
6-(piperidin-3-yl)-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)pyrimidin-4-amine
3-(1H-imidazol-1-yl)-6-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyridazine
2-(2-methoxypyridin-3-yl)pyridine-4-carboxamide
1-butyl-4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-2-one
methyl 3-[2-(2-fluorophenyl)acetyl]-9-[2-(morpholin-4-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(3,4-difluorophenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-(4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
N-benzyl-2-ethyl-4-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1,3-oxazole-5-carboxamide
N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-phenylpropanamide
2-(3-fluorophenoxymethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,3-oxazole-4-carboxamide
4-[2-chloro-4-(3-methoxypiperidine-1-carbonyl)phenoxy]-1-(2,2-dimethylpropyl)piperidine
3-{1-[(2-phenylpyrimidin-5-yl)methyl]piperidin-2-yl}propanoic acid
3-{[1-(1-methylpiperidine-4-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
(1R,5R)-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
N-cyclooctyl-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-[(2S,4R,6S)-2-ethyl-6-{2-[2-(piperidin-1-yl)ethoxy]phenyl}oxan-4-yl]acetamide
1-cyclopentyl-N5-[(4-methoxyphenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1'-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-chlorobenzamide
methyl 5-[3-(2-{[(3,4-difluorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]-5-oxopentanoate
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
1-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-4-benzyl-3-ethyl-1,4-diazepan-5-one
2-[(2R,3R)-2-hydroxy-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl]-3,5-dimethyl-1,4-dihydropyridin-4-one
N-(1H-imidazol-2-ylmethyl)-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
6-(2-hydroxyethyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-({1-[(4-acetamidophenyl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
N-[2-(2,3-dimethoxyphenyl)ethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S,4R)-1-benzyl-N,N-diethyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
3-ethyl-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-indole-2-carboxamide