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(2R,3R,6R)-3-(4-methoxyphenyl)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(4-fluorophenyl)-4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)[(2-methoxypyrimidin-5-yl)methyl]methylamine
N-[2-(4-fluorophenyl)ethyl]-9-methyl-10-oxo-3,9-diazaspiro[5.6]dodecane-3-carboxamide
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrazole-3-carbonyl)piperidine
9-(4-chloro-3-methylbenzoyl)-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
6-methoxy-N-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-(dimethylamino)-N-({2-[(dimethylamino)methyl]phenyl}methyl)-2-(2-fluorophenyl)acetamide
2,6-dimethyl-3-[4-(morpholine-4-carbonyl)piperazine-1-carbonyl]quinoline
2-amino-N,4-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-benzothiazole-6-carboxamide
[2-(3-methoxyphenyl)-1-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl](methyl)(pyridin-4-ylmethyl)amine
methyl 3-(2-chlorobenzamido)-5-{[3-(pyridin-3-yl)propanamido]methyl}benzoate
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(pyridin-3-yl)propanamide
4-cyclopropyl-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-4-methylpyrrolidin-2-one
5-({4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2-methoxyphenol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
5-(8-methoxy-2-methylquinolin-5-yl)pyridine-3-carboxamide
3-(3-hydroxyphenyl)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]propanamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-(1,3-dihydroxypropan-2-yl)-3-(2-fluorophenyl)benzamide
({4-[(2-fluoro-5-methylphenyl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
N-{3-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]phenyl}acetamide
2-ethyl-4-methyl-N-[1-(thiophen-2-yl)butyl]-1,3-oxazole-5-carboxamide
2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
1,4,6-trimethyl-N-{[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(1-{1-[(3-phenoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
1-(2-methoxyethyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-(2-{7-[(3-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
5-methyl-N-(pyridin-3-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-oxazole-4-carboxamide
1-[(4-phenyloxan-4-yl)methyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
2-methyl-3-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyrazine
({4-ethyl-5-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
[(1,2-dimethyl-1H-imidazol-5-yl)methyl]({[2-(2-methylphenoxy)pyridin-3-yl]methyl})amine
N,N-dimethyl-3-[({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}amino)methyl]pyridin-2-amine
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-phenylpropanamide
3-[6-(benzyloxy)pyridin-3-yl]-5,6-dimethyl-1,2-dihydropyridin-2-one
[1-(5-methyl-1,2,4-oxadiazol-3-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
3-[(3R,4S)-1-(isoquinolin-1-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-3-[(4-methoxyphenyl)methyl]-1,2-oxazole-5-carboxamide
4-{3-[4-(1-methoxypropan-2-yl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
6-(2-chlorophenyl)-2-[3-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butan-1-one
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[3-(methylsulfanyl)propyl]piperidine
2,6-difluoro-N-{[7-(3-phenylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-methylbutanamide
7-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-5-[2-(piperidin-1-yl)ethyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-N-[(2R)-3-methylbutan-2-yl]piperidine-1-carboxamide