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1-cyclohexyl-2-(furan-2-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-oxo-1-phenyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxamide
(3S)-4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-ethyl-3-methylpiperazin-2-one
4-ethyl-1-methyl-3-{1-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(4-chlorophenyl)methyl]-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine
2-[3-(dimethylamino)propyl]-9-[6-(methoxymethyl)pyridine-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(butylsulfanyl)-6-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]pyrimidin-4-amine
1-{2-methyl-4-[(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-[1-(2-methylbutanoyl)piperidin-4-yl]imidazolidine-2,4-dione
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2-methoxy-4-methylbenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yl)propyl]acetamide
N-[(3R,4S)-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3-methoxypropanamide
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
3-{3-methyl-5-[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
ethyl 4-(cyclopropylmethyl)-1-[1-(4-fluorophenyl)propan-2-yl]piperidine-4-carboxylate
6-(2,3-dimethoxy-5-methylphenyl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1-cyclopropyl-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-5-oxopyrrolidine-3-carboxamide
3-fluoro-4-methoxy-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
1-[2-({[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}(methyl)amino)ethyl]piperidin-2-one
[4-(2-phenylethyl)-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl]methanol
3-[2-(3,4-difluorophenyl)ethyl]-1-(2-ethoxyethyl)piperidine
3-(1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxopropan-2-yl)-2,3-dihydro-1,3-benzoxazol-2-one
6-fluoro-4-(oxan-2-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
(3S,9aR)-3-(4-aminobutyl)-8-(3-methylbutyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-ethyl-3-[(1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-(1H-indol-5-yl)urea
N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
methyl 6-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]pyrazine-2-carboxylate
3-(2,3-dihydro-1H-isoindol-2-yl)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]propan-1-one
4-(4-ethoxyphenyl)-2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazole
5-benzyl-3-[2-(pyrrolidin-1-yl)ethyl]-5-[1-(thiophene-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
5-[(3-hydroxypiperidin-1-yl)methyl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-oxazole-3-carboxamide
2-[3-(2-methoxyethyl)-5-(1-methoxypropyl)-1H-1,2,4-triazol-1-yl]acetic acid
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl]-6-methylpyrimidin-4-amine
1-(2-methylpyridin-4-yl)-4-(1H-pyrazole-4-carbonyl)-1,4-diazepane
N,N-dimethyl-4-({[3-(2-methylphenyl)phenyl]carbamoyl}amino)butanamide
1-(1,3-benzoxazol-2-yl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-amine
1-[2-methoxy-5-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide
4-(4-chlorophenyl)-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}butanamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-methylacetamide
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-5-(phenoxymethyl)-1H-pyrazole
(4aS,8aR)-N-benzyl-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}ethan-1-one
{1-[3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]piperidin-3-yl}methanol
2-[benzyl(methyl)amino]-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
(3R,5S)-N-cyclopentyl-1-(2-methylpropyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide