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4-[4-(2-chlorophenyl)piperidin-4-yl]-2-[3-(methoxymethyl)pyrrolidin-1-yl]pyrimidine
(6-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)methanol
4-{1-[4-(4-methylpiperazin-1-yl)benzoyl]piperidin-3-yl}pyrimidine
N5-cyclopropyl-N6-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-benzyl-3-(piperidin-4-yl)-1-(pyridin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-ethyl-2-methyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-1,3-thiazole-5-carboxamide
2-(3-methyl-1,2,4-oxadiazol-5-yl)-N-(6-phenoxypyridin-3-yl)piperidine-1-carboxamide
methyl 3-(4-{3-tert-butyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-1H-pyrazol-1-yl)propanoate
N2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N4,6-dimethylpyrimidine-2,4-diamine
(1S,6R)-9-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
3-[(3R,4S)-4-(dimethylamino)-1-(2-ethylbenzoyl)piperidin-3-yl]propan-1-ol
[(2,3-dimethoxyphenyl)methyl](methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-[2-(4-chlorophenyl)ethyl]-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-(pyrrolidine-1-carbonyl)pyridin-2-amine
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]quinoline-8-sulfonamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
2-{[4-(2-fluorophenyl)-5-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
[(3aS,6aS)-2-(2,6-dimethylquinoline-4-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methanol
N-tert-butyl-2-{[5-(pyrrolidin-2-yl)thiophen-2-yl]formamido}acetamide
3-({[2-(4-methoxyphenyl)ethyl]amino}methyl)-6-methyl-1-(prop-2-en-1-yl)-1,2-dihydroquinolin-2-one
methyl 5-(2-amino-5-methylpyrimidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2S)-N1-[4-(3-chlorophenyl)phenyl]-N2-ethylpyrrolidine-1,2-dicarboxamide
2-(1-benzylpiperidin-4-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
6-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrazine-2-carboxamide
{4-benzyl-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}methanol
N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-({7-[3-(trifluoromethyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
(3R,4R)-3-hydroxy-N-(2-methylphenyl)-4-{[2-(2-oxoimidazolidin-1-yl)ethyl]amino}pyrrolidine-1-carboxamide
2-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}-4,5,6,7-tetrahydro-1,3-benzothiazole
3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-(quinolin-3-ylmethyl)propanamide
(2,2-diphenylethyl)(methyl)[1-(pyrimidin-4-yl)ethyl]amine
4-(3-methylbutyl)-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
8-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-benzyl-1,3-thiazole-4-carbonyl)-1,2-oxazolidin-4-ol
3-(3,3-diphenylpiperidine-1-carbonyl)pyridin-2-ol
3-(hydroxymethyl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-3-ol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(4-methylpiperazin-1-yl)propanamide
(1R,5R)-6-(cyclopentylmethyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-3-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]urea
2-ethyl-N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
2-(2-fluorophenyl)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
4-(4-chlorophenyl)-1-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]butan-1-one
N'-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N'-methylethanediamide
5-ethyl-2-methyl-4-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
3-methyl-N-{[1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]methyl}but-2-enamide
1-[2-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one