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1-[4-(2-methylphenoxy)piperidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
methyl 4-[({[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)methyl]benzoate
9-[3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(methylamino)-1,3-thiazole-4-carboxamide
9-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
2,5-dimethyl-4-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidine
2-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxy-N-methyl-N-(propan-2-yl)pyrimidine-5-carboxamide
methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]{[2-(1H-pyrazol-1-yl)phenyl]methyl}amine
5-(1H-1,3-benzodiazol-2-ylmethyl)-1-methyl-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(hydroxymethyl)-2-methyl-4-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}methyl)pyridin-3-ol
1-[2-methoxy-4-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]azepan-3-amine
2-(2,5-dimethoxyphenyl)-N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}acetamide
N-[(3S,4R)-1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
8-[3-(thiophen-3-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(2-fluorophenyl)methyl]-N-(furan-3-ylmethyl)piperidin-3-amine
1-[4-({4-[3-(3-methylphenyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
7-(2,6-dimethoxyphenyl)-4-(4-fluorobenzoyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-chloro-4-(1-cyclobutyl-1H-imidazol-2-yl)phenol
N-[3-(3-methoxyphenyl)phenyl]-1-(3-methylbutyl)piperidine-4-carboxamide
methyl[(4-methyl-1H-imidazol-5-yl)methyl]{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
(3S,4R)-3-ethyl-4-methyl-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-ol
7-chloro-2-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1,3-benzoxazol-2-amine
(1H-imidazol-2-ylmethyl)(methyl){[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}amine
1-[4-ethoxy-3-(trifluoromethyl)phenyl]-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]urea
4-(3-methylpyridin-4-yl)-N-(1,3,4-thiadiazol-2-yl)-1,4-diazepane-1-carboxamide
3-chloro-5-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
3-[(4-fluorophenyl)methyl]-N-methyl-N-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
(1S,5R)-3-[(4-chlorophenyl)methyl]-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)acetamide
5-cyclopropanecarbonyl-1'-(5-propyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{1-benzyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}pyrazine
N-[3-(4-fluorophenyl)phenyl]-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxamide
1-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(pyridin-3-yl)ethan-1-one
methyl[(5-methyl-1H-pyrazol-3-yl)methyl]{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-(3-methylphenoxy)-1-[2-(pyridin-3-yl)acetyl]piperidine-4-carboxylic acid
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
N-(3-acetamido-4-methoxyphenyl)-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
2-methyl-N-[1-(6-methylpyridin-3-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-(benzenesulfonyl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
3-[2-(azocan-1-yl)-2-oxoethyl]-4-(furan-3-ylmethyl)piperazin-2-one
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[4-(hydroxymethyl)piperidin-1-yl]methyl}piperidin-2-one
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
N-[(2R,3R)-2-methoxy-1'-[(3-methylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
N-(furan-2-ylmethyl)-2-[3-(2-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-(prop-2-yn-1-yl)acetamide
3-(2-methoxyphenyl)-N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]propanamide
2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]benzonitrile
3-{methyl[3-oxo-3-(2-phenylazetidin-1-yl)propyl]amino}-1λ6-thiolane-1,1-dione