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methyl (2S,3S)-2-{[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-3-yl]formamido}-3-methylpentanoate
N3-[2-(adamantan-1-yl)propan-2-yl]-N5-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(3-methoxyphenyl)methyl]-N-methylacetamide
3-[(4-ethylphenyl)methyl]-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(piperidin-1-yl)piperidine
2,6-dimethyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]imidazo[1,2-a]pyridine-3-carboxamide
methyl 3-{4-[2-amino-3-cyano-6-(3-fluorophenyl)pyridin-4-yl]-1H-pyrazol-1-yl}propanoate
9-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[2-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
2-{[3-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[1,2-a]piperazine
8-(1H-imidazol-2-ylmethyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(3,4-dimethoxyphenyl)methyl]-4-{4-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[1-(1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
N-{2-[(3S)-3-hydroxypyrrolidin-1-yl]-2-oxoethyl}-N-(4-methylphenyl)methanesulfonamide
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-(3-hydroxy-3-methylbutyl)benzamide
2-cyclopentyl-N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
6-{[cyclopropyl(propyl)amino]methyl}-N-(1,4-dioxan-2-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(1S,5R)-6-benzyl-3-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(3S)-4-[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1-ethyl-3-methylpiperazin-2-one
1-(2-methyl-1,3-thiazole-5-carbonyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
2-(cyclopropylmethyl)-8-[4-(1H-imidazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
8-[5-(4-chlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[(5-methylpyrazin-2-yl)methyl]acetamide
1-cyclohexyl-4-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
4,6-dimethyl-N-[3-(propan-2-yloxy)propyl]quinazolin-2-amine
(2R,6R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{1-[1-(4-formylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-2,3-dihydro-1-benzofuran-7-carboxamide
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-(2-phenylpropyl)piperidine-4-carboxamide
N4-cyclopropyl-6-{4-[(2-ethylpyrimidin-5-yl)methyl]piperazin-1-yl}pyrimidine-2,4-diamine
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-(2-methylpropyl)pyrrolidin-2-one
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-propoxypiperidine
2-hydroxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(methylsulfanyl)butanamide
3-[(6-hydroxy-1,4-oxazepan-4-yl)sulfonyl]-N-phenylbenzamide
3-[methyl({5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl})amino]propanamide
7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[3-(2-methoxybenzoyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(5S,9aS,9bS)-5-(4-chlorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(2-fluoro-3-methoxyphenyl)pyridine
1-(2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
(2S)-3-(4-hydroxyphenyl)-2-{[3-(1H-imidazol-2-yl)phenyl]formamido}propanamide
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-2,3-dihydro-1,2-benzothiazol-3-one
2-({4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one