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N-methyl-N-[(4-methyl-1H-imidazol-5-yl)methyl]-2,3-dihydro-1H-inden-2-amine
6-(cyclopropylmethoxy)-4-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-(2-methylphenyl)-1,2,4-triazin-3-amine
3-(1-cyclohexanecarbonylpiperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
3-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidine-1-carbonyl]-2H-chromen-2-one
9-methoxy-3-{[1-(propan-2-yl)-1,2,3,4-tetrahydroquinolin-6-yl]methyl}-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
methyl 3-(2,2-dimethyloxane-4-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-oxo-8-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(dimethyl-1,2-oxazol-4-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
2-methyl-4-phenyl-9-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-(2-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
3-[3-({[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
3-phenyl-N-(4-{4-[(quinolin-6-ylmethyl)amino]piperidin-1-yl}phenyl)propanamide
(4aS,8aR)-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
6-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[3-(4-fluorophenyl)propyl]oxane-4-carboxamide
6-[(3,5-dimethoxyphenyl)methoxy]-1-(propan-2-yl)-4-[2-(pyridin-2-ylsulfanyl)acetyl]-1,4-diazepan-2-one
N-({7-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
2-(3,4-dichlorophenyl)-4-(2,5-dimethylpyrimidin-4-yl)morpholine
N-(1H-imidazol-2-ylmethyl)-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
(4aS,7aR)-1-[(4-acetylphenyl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1-benzothiophene-5-carboxamide
4-(2-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,3-thiazol-2-amine
N-(3-ethoxypropyl)-3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(2-methylpropyl)piperidin-3-yl]propanamide
1-[4-(2-{[cyclohexyl(methyl)amino]methyl}quinazolin-4-yl)piperazin-1-yl]ethan-1-one
1-[2-({[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]propan-1-one
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidine
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-methoxyethan-1-one
6,7-dimethoxy-3-(thiophen-2-ylmethyl)-3,4-dihydroquinazolin-4-one
2-(1-methyl-1H-pyrrol-3-yl)-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]acetamide
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-4-(methylsulfanyl)benzamide
methyl 9-(cyclopentyloxy)-7-oxo-3-(pyridin-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopent-1-ene-1-carboxamide
3-(methoxymethyl)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,2,4-triazole
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-(thiophen-3-ylmethyl)propanamide
1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-ethylpiperazine
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]propanamide
N-{3-oxo-3-[4-(propan-2-yl)piperazin-1-yl]propyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
methyl (2S)-1-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}pyrrolidine-2-carboxylate
1-(4-fluoro-2-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}phenyl)-1H-pyrazole
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(1H-imidazol-4-yl)-2-(1H-pyrrol-1-yl)propan-1-one
2-(oxolan-3-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
1-(2,4-difluorophenyl)-5-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethyl)-1H-1,2,4-triazole
2-[methyl(1,3-thiazol-2-ylmethyl)amino]-2-{4-[(morpholine-4-carbonyl)amino]phenyl}acetic acid
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(pyridin-2-yl)ethyl]amino}methyl)piperidin-2-one
propan-2-yl 3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxylate
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide
N-[2-(4-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]methanesulfonamide