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5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(thiophene-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
4-benzyl-1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-ethyl-1,4-diazepan-5-one
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-(1-methyl-5-oxopyrrolidin-3-yl)urea
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[2-(3-methoxyphenyl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-(2-methyl-1H-pyrrole-3-carbonyl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(cyclopropylmethyl)-4-(3-phenyl-1H-pyrazole-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
2-{[1-(3-hydroxybutyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
4-(1-benzothiophen-2-ylmethyl)-11-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(2-methylphenyl)methyl]-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-1,2,3-triazole
1-{2-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
N-[2-(dimethylamino)ethyl]-3-[5-(2,2-dimethylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
(1R,2R,6S,7S)-4-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-{1-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]piperidin-3-yl}benzoic acid
3-(ethylsulfanyl)-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(3-methoxypropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-methoxyethyl)-1-[1-(4-methylbenzoyl)piperidin-4-yl]piperidine-3-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(1-methyl-1H-1,2,4-triazol-5-yl)-1H-pyrazol-1-yl]acetamide
1-(4-ethoxyphenyl)-2-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[1-(pyridin-3-yl)propan-2-yl]amine
6-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)[(3-phenoxyphenyl)methyl]amine
2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}thiophene-3-sulfonamide
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
methyl({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
2-[3-(1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyrazine
N-{[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]methyl}quinoline-5-carboxamide
2-{4-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
2,3-dimethyl-N-[2-(pyridin-3-yl)ethyl]quinoxaline-6-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-(butan-2-yl)-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-yl)-3-phenylpropan-1-ol
methyl (1R,3S,3aR,6aS)-3-[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
5-[1-(1H-imidazol-4-ylmethyl)pyrrolidin-2-yl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]thiophene-2-carboxamide
1-benzyl-3-(2-methoxyethyl)-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-(pyrazin-2-ylmethyl)acetamide
(3S)-4-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1-ethyl-3-methylpiperazin-2-one
1-ethyl-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propane-1-sulfonamide
1-[6-(2-methoxyphenyl)pyridazin-3-yl]-3-phenylpyrrolidin-3-ol
3-{[(furan-3-ylmethyl)(methyl)amino]methyl}-N-(1-methyl-1H-imidazol-2-yl)benzamide
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-[(2-phenoxypyridin-3-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-methyl-2-[(4-methylphenyl)amino]-2-phenylpropanamide
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(pyridin-4-yl)propan-1-one
(3S,4R)-4-(3-fluorophenyl)-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidine-3-carboxylic acid
3-ethyl-5-{1-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2-oxazole
1-[2-(diethylamino)acetyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-[2-(2-chloropyridine-4-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-6-methylpyridine
(1R,5R)-N,N-dimethyl-6-[(5-propylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide