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4-phenyl-N-(1-{1-[3-(pyridin-4-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
3-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-3,9-diazaspiro[5.5]undecane
3-(1H-pyrazol-1-ylmethyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]benzamide
2,6-diamino-4-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(2S)-4-methyl-2-[(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}phenyl)formamido]pentanamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-{[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]methyl}furan-2-carboxamide
N-[2-(diethylamino)ethyl]-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonane-7-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
5-[1-(3,5-difluorobenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3,4-dihydropteridin-4-one
(1R,5S,8S)-3-{[3-(methylsulfanyl)phenyl]methyl}-3-azabicyclo[3.2.1]octan-8-ol
5-[({[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-1,3-benzodiazole-7-carboxamide
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-(quinolin-6-ylmethyl)propanamide
N-[(2-chloro-3,4-dimethoxyphenyl)methyl]-N-methyloxan-4-amine
1-{5-[(1E)-pent-1-en-1-yl]-1H-1,3-benzodiazol-2-yl}ethan-1-ol
2-[3-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]acetamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(5-oxo-1-phenylpyrrolidin-3-yl)acetamide
2-cyclopentyl-9-[(5-methylfuran-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-8-[2-oxo-2-(piperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3R,4R)-1-(2,5-dimethylpyrimidin-4-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
N-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
3-{[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)amino}-1-phenylpropan-1-ol
2-(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
3-methanesulfonyl-N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
N-(2-methyl-1-benzofuran-5-yl)-3-(pyrimidin-4-yl)piperidine-1-carboxamide
N-{1-[1-(3-chlorobenzoyl)piperidin-4-yl]-2-(2,4-difluorophenyl)ethyl}-N-methylpropanamide
(2S,4R)-4-(2-cyclopentylacetamido)-N-(isoquinolin-5-ylmethyl)-N-methylpyrrolidine-2-carboxamide
1-({1-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-yl}methyl)pyrrolidin-2-one
N-[(2S)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
N-(6-hydroxy-6-methylheptan-2-yl)-5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
4-(1-hydroxy-2-{4-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-1,2,3-triazol-1-yl}ethyl)phenol
methyl({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})(thiophen-3-ylmethyl)amine
{4-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
4-(3-benzyl-1H-pyrazol-5-yl)-1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidine
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
ethyl 1-[3-(furan-2-yl)propanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
2,3-dimethyl-7-{1H-pyrrolo[2,3-c]pyridin-5-ylmethyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-{1-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}-5-ethylpyridine
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-5-methyl-3-phenyl-1,2-oxazole
1-(2-oxo-2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-1,2-dihydroquinoxalin-2-one
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(3-methylpyridin-2-yl)ethyl]benzamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
1-{2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}pyrrolidin-2-one
(3S,4R)-3-methoxy-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-4-amine