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7-[(4-fluorophenyl)methyl]-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decane
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(4-fluoro-3-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-(4-methyl-6-{[3-(4H-1,2,4-triazol-4-yl)propyl]amino}pyrimidin-2-yl)phenol
1-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}azetidin-3-ol
1-{7-[1-(dimethylamino)-2-hydroxypropan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
1-[(5-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}-2-methoxyphenyl)methyl]-1H-pyrazole
(3S,4R)-4-(4-fluorophenyl)-1-(4-hydroxy-1-methylpiperidine-4-carbonyl)pyrrolidine-3-carboxylic acid
2-{3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-N-(furan-2-ylmethyl)acetamide
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-2-(1,2,3,6-tetrahydropyridin-4-yl)ethan-1-one
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
1-[4-(4-methylphenyl)-5-(pyridin-4-yl)pyrimidin-2-yl]piperidine-3-carboxamide
1-(2-{[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
[3-(2-methoxyethyl)-1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl]methanol
methyl 2-(3-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}-1H-indol-1-yl)acetate
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-propylpiperidin-4-yl)acetamide
3-{5-[3-(2-methoxyphenyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
ethyl 4-[1-(5-fluoro-1H-indole-2-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
1-(5-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(piperidin-1-yl)propan-2-ol
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
4-[(3,5-dichloro-4-methylphenyl)formamido]-N,4-dimethylpentanamide
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]propanamide
N-cyclohexyl-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-(2-phenylethyl)acetamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl){[4-(methylsulfanyl)phenyl]methyl}amine
(3S,4S)-4-(3-methoxyphenyl)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
N3-[1-(2-chlorophenyl)ethyl]-N5-cyclooctyl-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-amino-6-(2-methylpropanoyl)-4-[2-(propylamino)pyrimidin-5-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-{1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
6-(2-aminoethyl)-N-(cyclopropylmethyl)-N-propylpyrimidin-4-amine
2-methoxy-4-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(2-methoxyethyl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
1-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}naphthalen-2-ol
3-(4-methanesulfonylphenyl)-5-methoxypyridine
1-(ethanesulfonyl)-3-[2-(methylsulfanyl)benzoyl]piperidine
ethyl 5-[(3-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-({7-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
3-{4-[(1-butyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
5-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
1-{1-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperidin-4-yl}butan-1-one
1-[2-(methylamino)pyridine-3-carbonyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)-3-(pyridin-3-yl)propan-1-one
methyl 1-({4-[2-(4-chlorophenyl)acetyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
7-(3-chlorophenyl)-4-(quinolin-6-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 4-[2-(1-methyl-3-oxopiperazin-2-yl)acetamido]piperidine-1-carboxylate
methyl 3-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}benzoate
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
3-{4-[(6-methoxypyridin-3-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
3-acetamido-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(3-fluoro-4-methylphenyl)methyl]piperidine-3-carboxamide
1-[2-(2-phenylethyl)morpholin-4-yl]pent-4-en-1-one
1-{3-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}imidazolidin-2-one