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5-[(4-ethylpiperazin-1-yl)methyl]-N-(3,3,5,5-tetramethylcyclohexyl)-1,2-oxazole-3-carboxamide
1-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]ethyl}-3-(2-ethoxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-{2-[5-(1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine-4-carboxamide
6-oxo-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1,6-dihydropyrimidine-5-carboxamide
6-fluoro-2-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)quinolin-4-ol
N-benzyl-2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
7-methanesulfonyl-4-methyl-2-[4-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]quinazoline
4-chloro-1-ethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-3-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
5-[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
5-{2-[4-(2-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-(1H-imidazole-2-carbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[3-({[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]carbamoyl}amino)phenyl]butanamide
3-(1-butanoylpiperidin-4-yl)-N-cyclopropylpropanamide
N-methyl-N-{2-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}methanesulfonamide
N-[1-(2-chlorophenyl)ethyl]-3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-9-(3,3,3-trifluoropropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-cyano-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]cyclopropane-1-carboxamide
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
2,3,5,6-tetramethyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]benzamide
2-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
1-[(2-fluorophenyl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-[2-(2-fluorophenyl)ethyl]-1-(furan-2-carbonyl)piperidine
1-(7-methoxy-4-methylquinazolin-2-yl)-N-[(3-methylphenyl)methyl]piperidine-3-carboxamide
N-(2-hydroxypropyl)-2-[5-oxo-3-phenyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-4-sulfamoylbenzamide
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}benzenesulfonamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[phenyl(pyridin-4-yl)methyl]propanamide
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-1-methyl-4-oxo-N-(pyridin-3-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
1-(2-ethoxyethyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}phenol
3-(3-{[ethyl(oxan-2-ylmethyl)carbamoyl]amino}phenyl)-N,N-dimethylpropanamide
N,N-dimethyl-2-{3-oxo-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-4-yl}ethane-1-sulfonamide
methyl (1R,3S,3aR,6aS)-3-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-(1-{[1-(3-methylbutyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
methyl[(1-phenylpyrrolidin-3-yl)methyl]{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
8-fluoro-3-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-1,4-dihydroquinolin-4-one
2-(5-methyl-4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1H-pyrazol-1-yl)-4-(5-methylfuran-2-yl)pyrimidine
(2S,4R)-4-amino-N-methyl-1-[(2,4,6-trimethylphenyl)methyl]pyrrolidine-2-carboxamide
3-chloro-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-2-methyl-N-(pyridin-3-ylmethyl)benzene-1-sulfonamide
5-benzenesulfonamido-1-ethyl-2-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[4-(morpholin-4-yl)butyl]acetamide
2-(4-{[3-(2-methylphenyl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
3-methoxy-N,4-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]benzamide
1-(3-chlorophenyl)-5-methyl-4-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]piperazin-2-one
3-(3,4-difluorophenyl)-5-(4-methyl-1H-imidazol-2-yl)-1,2,4-oxadiazole