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5-fluoro-2-(1-{1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)-1H-1,3-benzodiazole
N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
ethyl 1-{[2-(2-hydroxyethoxy)phenyl]methyl}-3-(2-phenylethyl)piperidine-3-carboxylate
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
4-(4-chlorophenyl)-N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}butanamide
N-{[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]methyl}furan-2-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
3-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
3-{1-[1-(furan-3-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
3-[(3-methoxyphenyl)methyl]-8-[(4-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(2S,4R,5R)-4-[({[3-(ethoxymethyl)-4-methoxyphenyl]methyl}amino)methyl]-5-(2-fluorophenyl)-1-methylpyrrolidin-2-yl]methanol
(1S,5R)-3-[(4-chloro-2-fluorophenyl)methyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[5-(methoxymethyl)thiophene-2-carbonyl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-(1-{7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
2-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)-1-methyl-1H-imidazole
3-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(prop-2-en-1-yl)propanamide
N-methyl-3-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-hydroxyethyl)-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
N-[1-(1-cyclopropylethyl)-1H-pyrazol-5-yl]-2-[5-(1H-pyrazol-3-yl)-1H-indol-1-yl]acetamide
2-ethyl-9-[5-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-({7-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-phenylmethanesulfonamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(4-hydroxyphenyl)propyl]acetamide
2-(2-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenoxy)ethan-1-ol
1-(cyclohexylmethyl)-N-[(1-hydroxycyclohexyl)methyl]-6-oxopiperidine-3-carboxamide
(3S,4S)-4-(propan-2-yloxy)-1-(2,6,8-trimethylquinoline-4-carbonyl)pyrrolidin-3-ol
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]urea
4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(propan-2-yl)piperidine
3-(4-hydroxyphenyl)-N-{3-[(pyridin-3-yl)amino]propyl}-1H-pyrazole-5-carboxamide
1-{2-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}-1,3-diazinane-2,4-dione
N-[4-(methylsulfanyl)phenyl]-6-(2-phenoxyacetyl)-6-azaspiro[2.5]octane-1-carboxamide
(3R,4R)-4-cyclopropyl-1-(6-cyclopropylpyrimidin-4-yl)-3-methylpiperidin-4-ol
(2S,4R)-1-[(3,5-dimethoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N-[1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]-N-methylacetamide
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-[4-(4-fluorophenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-[(2-fluorophenyl)methyl]acetamide
4-methyl-N-[1-(thiophen-2-yl)propan-2-yl]-1,3-oxazole-5-carboxamide
4-{[3-(3-{furo[3,2-c]pyridin-4-yl}phenyl)-1H-pyrazol-1-yl]methyl}-1,3-thiazole
4-(cyclopropylmethyl)-N-(2-methoxyphenyl)-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
5-cyclopropanecarbonyl-1'-(4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{[(3S,4R)-1-[(2-ethylphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-[(3,4-difluorophenyl)methyl]-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[3-(propan-2-yloxy)propyl]piperidine-4-carboxamide
3-(5-{[(oxolan-2-ylmethyl)carbamoyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(pyrrolidin-1-yl)ethyl]amine
2-{[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(2-methylphenyl)methyl]amino}ethan-1-ol
N-(2-methyl-1,3-benzothiazol-5-yl)-6-(thiolan-3-yl)-6-azaspiro[2.5]octane-1-carboxamide
1-[5-(1-ethylpiperidin-4-yl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-3-ol
5-(1-cyclopentyl-1H-pyrazol-3-yl)-N-[(4-fluoro-3-methoxyphenyl)methyl]-4-methyl-1,3-thiazol-2-amine