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N-[1-cyclopentyl-7-(morpholine-4-carbonyl)-1H-1,3-benzodiazol-5-yl]benzamide
N-{1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylpyridine-3-carboxamide
1-(1-{2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetyl}piperidin-4-yl)-1,4-diazepan-5-one
(4aS,8aR)-6-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(4-ethylpiperazin-1-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-benzofuran-2-carboxamide
N-(3-methylphenyl)-3-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]propanamide
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methyl-N-(propan-2-yl)acetamide
1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
1-{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}piperidin-3-amine
methyl 2-{[(3S,4R)-3-acetamido-4-propylpyrrolidin-1-yl]sulfonyl}benzoate
4-[1-(3-chloro-4-methylphenyl)piperidin-4-yl]-N,N-dimethylmorpholine-2-carboxamide
N-[2-(dimethylamino)ethyl]-5-methyl-6-(morpholine-4-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-(2-{2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)acetamide
7-methoxy-3-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
2-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-N-ethylacetamide
N-(5-hydroxyadamantan-2-yl)-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carboxamide
1-cyclopropyl-3-(2-{4-[(3-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
3-(4-methyl-1,3-thiazol-5-yl)-1-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}propan-1-one
3-{[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl](pyrrolidin-1-yl)methyl}pyridine
methyl (2S,4R)-1-(propan-2-yl)-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
[2-(dimethyl-1,3-thiazol-2-yl)ethyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
methyl 9-[(4-fluorophenyl)methoxy]-7-oxo-3-(pyridin-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[1-(6-methylquinoline-4-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
4-(3,4-dimethoxybenzoyl)-1-(2-methylphenyl)piperazin-2-one
1-(cyclohexylmethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-({5-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}methyl)pyridine
N-[4-({methyl[1-(1,2-oxazol-3-yl)ethyl]carbamoyl}methyl)phenyl]butanamide
N,N-dimethyl-2-[(1S,5R)-6-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
4-(4-{[2-(1H-indol-1-yl)ethyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
N-(2,4-dimethylphenyl)-2-[(2-phenylpropyl)amino]acetamide
methyl 4-{[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazol-4-yl]formamido}butanoate
3-{5-[(2,2,6,6-tetramethylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,4-dihydroquinolin-4-one
5-ethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]pyrimidin-2-amine
2-chloro-N-[1-(1-cyclopentylpiperidin-4-yl)-1H-pyrazol-5-yl]benzamide
2,3,5-trimethyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-fluoro-4-hydroxy-N-methyl-N-[2-(oxan-2-yl)ethyl]benzamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrrolidine-1-sulfonamide
3-[(4aR,7aS)-4-(6-aminopyridine-3-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
8-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}quinoline
1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-methanesulfonyl-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidine-2-carboxamide
4-fluorophenyl (7S,9aR)-7-(hydroxymethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
4-[3-(2-methyl-1,3-thiazol-4-yl)-1-phenyl-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
(4aS,7aR)-1-(2-methoxybenzenesulfonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-chloro-2-methylbenzoyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine
3-(naphthalene-2-sulfonyl)-3,9-diazaspiro[5.6]dodecan-10-one