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N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
9-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(2-methyl-1,3-thiazol-4-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
1-{3-[4-(4-methoxyphenyl)-2-methylpiperazine-1-carbonyl]phenyl}imidazolidin-2-one
1-cyclopentyl-4-(7-fluoroquinazolin-4-yl)piperazin-2-one
4-[4-(2-methoxyphenoxy)piperidin-1-yl]-5,6-dimethylpyrimidine
1-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
methyl (2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-[(pyridin-2-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-(9H-purin-6-yl)piperidin-4-amine
1-[(2S,4S)-1-[(4-methoxynaphthalen-1-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
3-{1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-N-phenylpropanamide
1-(4-benzylpiperidin-1-yl)-3-[1-(1H-imidazole-4-carbonyl)piperidin-4-yl]propan-1-one
2-{2-[(3-chlorophenyl)methoxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-methoxy-4-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,3-thiazole-5-carboxamide
2-(4-chlorophenyl)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-hydroxyethan-1-one
methyl 6-(1-benzofuran-2-carbonyl)-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-methyl-2-(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
N-(1,3-benzothiazol-2-yl)-3-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]propanamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(quinolin-5-ylmethyl)acetamide
2-cyclopentyl-9-(pyrimidin-5-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-tert-butylphenyl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
(3aS,7aR)-2-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-(3-hydroxypropyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyridin-2-yl)ethan-1-one
[4-(2-phenoxyethyl)-1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl]methanol
2-[2-(4-fluorophenyl)morpholin-4-yl]-1,3-thiazole-4-carboxamide
(3S)-3-methyl-1-(2-methylpropyl)-4-{2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperazin-2-one
1-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
(1R,5R)-3-cyclobutanecarbonyl-6-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-N-methyl-3-(propan-2-yl)-N-(quinolin-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}propanamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(1H-pyrazol-4-yl)butanamide
N-methyl-2,3-dioxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(6-hydroxy-6-methylheptan-2-yl)-5-methyl-1H-pyrazole-4-carboxamide
2-methoxy-4-methyl-N-(1,4-oxazepan-6-ylmethyl)benzene-1-sulfonamide
2-(4-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzoyl}piperazin-1-yl)pyrimidine
1-methyl-3-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
methyl 6-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
2-chloro-4-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
3-benzyl-4-(4-chlorobenzoyl)piperazin-2-one
1-[2-(piperidin-2-yl)ethyl]-N-(pyrimidin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-(cyclohex-1-ene-1-carbonyl)-1-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-amine
1-({4-[(dimethyl-1H-1,2,4-triazol-3-yl)carbamoyl]phenyl}methyl)-N-methylpyrrolidine-3-carboxamide
1-methyl-3-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}methyl)-1,2-dihydroquinolin-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-[(3S,4R)-4-(dimethylamino)-1-(2,2-diphenylethyl)piperidin-3-yl]propanamide