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4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}benzamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(pyridin-2-yl)propanamide
N-(3,4-difluorophenyl)-6-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
6-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-methyl-1,3-benzothiazole
N-(butan-2-yl)-3-(1-methyl-1H-pyrrol-2-yl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
1'-[(5-methylthiophen-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl][(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amine
2-(cyclopropylmethyl)-7-[2-(ethylamino)pyrimidine-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[3-(propan-2-yloxy)propyl]benzamide
4-[(4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}furan-2-yl)methyl]morpholine
(3aS,6aS)-1-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-octahydropyrrolo[2,3-c]pyrrole
N-[(2R,3R)-1'-[(3-methoxyphenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,2-dimethyl-2-(thiophen-2-ylformamido)propanamide
1-[7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4-methylphenyl)propan-1-one
2-[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyrazine
N-(6-chloropyridin-3-yl)-8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
1-(2-{1-[(2R)-2-amino-3-(4-chlorophenyl)propanoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
2-(benzyloxy)-N-[(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)methyl]acetamide
2-chloro-N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)pyridine-4-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
methyl (2S)-2-({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)-2-phenylacetate
1-(2,2-dimethylpropyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-{4-[(6-fluoroquinolin-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
5-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]pyrrolidin-2-yl}-N-[2-(methylsulfanyl)ethyl]thiophene-2-carboxamide
2-(cyclopentylmethyl)-N-cyclopropyl-6-methyl-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
1-(2-aminoethyl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxy-1-oxopropan-2-yl}acetamide
N-(3-cyclopentylpropyl)-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
5-(morpholin-4-ylmethyl)-8-{[4-(trifluoromethyl)pyridin-2-yl]oxy}quinoline
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-{[(2S)-oxolan-2-ylmethyl]sulfamoyl}benzamide
2-[4-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]-1-(piperidin-1-yl)ethan-1-one
(1R,3s,6r,8S)-4-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
N-cyclooctyl-5-(3-methylpiperidine-1-carbonyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(1R,5R)-6-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(2,6-dichlorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1'-(2-methoxypyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-(cyclopropylmethyl)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine-3-carboxylic acid
3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-methyl-N-(thiophen-3-ylmethyl)propanamide
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-5-phenyl-1H-pyrrole-2-carboxamide
N-(1-hydroxy-3-methylbutan-2-yl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
1-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N,N-diethylpyrrolidin-3-amine
N-(3-hydroxybutyl)-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl}ethan-1-ol
N-[(2-chlorophenyl)methyl]-7-fluoro-N-(2-hydroxyethyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-(2-methoxyethoxy)-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
(1R,3S)-7-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-7-azaspiro[3.5]nonane-1,3-diol