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N-[1-(furan-2-yl)ethyl]-9-methoxy-3-[2-(3-methoxyphenyl)acetyl]-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)pyrrolidin-3-ol
5-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
2,5-dimethyl-3-(3-{1-[(6-methylpyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
2-(ethylamino)-N-(furan-2-ylmethyl)-N-(2-phenylethyl)pyrimidine-5-carboxamide
ethyl 5-methyl-3-[(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)formamido]hexanoate
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
N-(3-methylphenyl)-3-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}propanamide
1'-cyclopentanecarbonyl-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{imidazo[1,2-a]pyridin-2-yl}-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
methyl (2S,4R)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-(2,2-diphenylacetamido)pyrrolidine-2-carboxylate
(1S,4R)-1-[3-(3-chloro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]-4,7,7-trimethyl-2-oxabicyclo[2.2.1]heptan-3-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)[(5-methylfuran-2-yl)methyl]amine
1-[(2-ethoxyphenyl)methyl]-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
N-[2-(benzyloxy)ethyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
2-{2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}cyclopentan-1-one
4-{2-oxo-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperazin-1-yl}benzonitrile
3-{1-[2-(2H-indazol-2-yl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
3-{2-[(4aS,8aR)-1-(2-methylpropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-methylpiperazine
3,3-dimethyl-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
4-chloro-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[(4-methoxy-3-methylphenyl)methyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
1-(cyclopropylmethyl)-5-[(diethylcarbamoyl)methyl]-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-9-oxo-N-(propan-2-yl)-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-[2-(4-chlorophenyl)ethyl]-5-(2-{[(3-methylphenyl)methyl]amino}ethyl)pyrrolidin-2-one
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidine
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[3-(methylsulfanyl)propyl]piperidin-3-yl}propanamide
N-[4-(1H-indazol-1-yl)-2-methoxyphenyl]acetamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
methyl 2-(cyclopentylsulfamoyl)-6-[(2,3-difluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(3-{4-[(2-ethylbutanamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-5-methylthiophene-2-carboxamide
1-methyl-3-(propan-2-yl)-5-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-pyrazole
1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
2-fluoro-N-[3-oxo-3-(3-propylmorpholin-4-yl)propyl]benzamide
1-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]-4-phenylbutane-1,4-dione
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[(1-methylpiperidin-4-yl)methyl]amine
7-methoxy-3-{[4-(oxolan-2-ylmethyl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
(1S,9S)-11-(3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
1-ethyl-5-(4-fluoro-2-methoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
1-(furan-3-ylmethyl)-4-[2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
N-methyl-2-[2-oxo-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propanamide
N-benzyl-5-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
N,N,5-trimethyl-2-(quinolin-8-yl)pyrimidin-4-amine
(3S,4R)-1-{[3-(2-hydroxyethoxy)phenyl]methyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopentanecarboxamide