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N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(pyridin-2-yl)propanamide
4-(dimethyl-1,2-oxazol-4-yl)-3-(3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-ethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(2-chlorophenoxy)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-{4-[6-(methoxymethyl)pyrimidin-4-yl]piperazin-1-yl}pyridine-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[4-(morpholine-4-carbonyl)pyridin-2-yl]pyrrolidin-3-amine
2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
ethyl 1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[(2S,4R,6S)-2-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-6-(2-methylpropyl)oxan-4-yl]acetamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}propanamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[1-(pyridin-3-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
(2S,4R)-4-(cyclooctylamino)-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
5-(3-fluoro-4-methoxyphenyl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
1-[(3R)-3-hydroxy-3-phenylpropyl]-2-methyl-1,4-dihydroquinolin-4-one
2-(4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
1-(2,6-difluorobenzoyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
(1S,5R)-3,6-bis[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]-2-(trifluoromethyl)benzamide
2-{3-methyl-5-[3-(piperidine-1-carbonyl)pyrazin-2-yl]-1H-1,2,4-triazol-1-yl}acetic acid
6-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-(4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)propan-1-ol
1-benzyl-5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]azepane-4-carboxamide
N'-(butan-2-yl)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-N'-(3-phenylprop-2-yn-1-yl)ethanediamide
[2-(2,4-dimethylphenoxy)ethyl](methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
2-(3-fluoro-4-methoxybenzenesulfonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N,N-bis(prop-2-en-1-yl)propanamide
2-butyl-5-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}-1,3-benzoxazole
(3S,4R)-N,N-dimethyl-1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-amine
8-[(4-methoxy-2,3-dimethylphenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-ethyl-3-methyl-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}piperidine-3-carboxamide
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxylate
2-({1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}propan-1-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-(2-oxopyrrolidin-1-yl)acetamide
4-({4-[3-(2,2-dimethylpyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
2-{1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
2-(4-methoxyphenyl)-5-{[4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}pyrimidine
1-(2-benzyl-1,3-thiazole-4-carbonyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
{1-[(2,5-dimethoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
2-{1-[(5-methylfuran-2-yl)methyl]-4-[(2,4,5-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-fluoro-2-[3-(pyridin-3-yl)azetidin-1-yl]-4-(pyrrolidin-1-yl)pyrimidine
1-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)-3-propylpiperidine-3-carboxylic acid
1-(2-methyloxolane-2-carbonyl)-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[1-(1-phenylethyl)-1H-pyrazol-5-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
ethyl 4-{[4-(2-methoxy-2-phenylacetyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
1,3,7-trimethyl-2-(thiomorpholine-4-carbonyl)-1H-indole