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2-hydroxy-N-[2-(4-methylmorpholin-2-yl)ethyl]-5-(1H-pyrrol-1-yl)benzamide
6-methyl-4-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
7-cyclopropanecarbonyl-N-methyl-N-(oxan-2-ylmethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3S,4R)-4-(2-methylphenyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
3-(benzylsulfanyl)-1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}propan-1-one
3-{2-[4-(4-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-(2,3-dimethoxyphenyl)-4-(trifluoromethyl)pyrimidine
(1R,3S)-7-(6-aminopyridine-3-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
N-({8-cyclopropanecarbonyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(3,4-dimethoxyphenyl)acetamide
(1R,5R)-N,N-dimethyl-6-(quinolin-5-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(3R,5S)-5-(3-fluorophenoxymethyl)-N-(2-phenylethyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
2-{4-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]piperidin-1-yl}pyrimidine
2-(2-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}phenoxy)ethan-1-ol
N-[(2S,4R,6S)-2-(2-methylpropyl)-6-[4-(methylsulfamoyl)phenyl]oxan-4-yl]acetamide
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
2-methoxy-N-[(2R,3R)-1'-[(3-methylphenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
4-(4-methoxyphenoxy)-1-(oxane-4-carbonyl)piperidine
N-[2-(4-fluorobenzenesulfonyl)ethyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[(4-methoxyphenyl)methyl]-4-(thiophene-2-sulfonyl)morpholine
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
methyl 4-[({2-[1-(6-hydroxy-6-methylheptan-2-yl)-5-oxopyrrolidin-2-yl]ethyl}amino)methyl]benzoate
3-chloro-4-fluoro-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-3,4-dimethoxy-N-(oxolan-2-ylmethyl)benzamide
N-[2-(2,4-difluorophenyl)-1-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}ethyl]-N-methylcyclopropanecarboxamide
(5S,9aS,9bS)-5-[4-ethoxy-3-(hydroxymethyl)phenyl]-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
{1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-yl}methanol
N-cyclohexyl-3-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]propanamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(thiophen-3-ylmethyl)amino]pyrrolidin-2-one
dimethyl(1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]phenyl}ethyl)amine
2-chloro-N-{[1-(2-oxo-2-phenylacetyl)piperidin-3-yl]methyl}benzamide
ethyl 1-(4-oxo-3,4-dihydrophthalazine-1-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
4-(2-methoxyphenyl)-2-methyl-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazine
(5S,9aS,9bS)-5-(1-benzothiophen-2-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
6-{4-[1-(dimethylamino)ethyl]piperidin-1-yl}-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
methyl 4-({[(3R,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(methylcarbamoyl)pyrrolidin-3-yl]amino}methyl)benzoate
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
3-{[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]methyl}-N-methylbenzamide
N-[3-({3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}sulfonyl)phenyl]acetamide
5,7-dimethyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]pyrido[2,3-d]pyrimidin-4-amine
2-(dimethylamino)-N-{3-[1-(pyridin-2-ylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]propyl}acetamide
(2E)-N-cyclopropyl-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}-3-(thiophen-2-yl)prop-2-enamide
N-(3-hydroxypropyl)-4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]ethan-1-one
(1-{4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carbonyl}piperidin-2-yl)methanol
N-{[1-(carbamoylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-2-phenoxyacetamide
2-({4-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
(3S,4R)-3-benzyl-1-[(2-fluoro-3-methoxyphenyl)methyl]-4-methylpiperidin-4-ol
methyl 1-[6-oxo-1-(3-phenylpropyl)piperidine-3-carbonyl]piperidine-4-carboxylate